Structure-guided design of potent and selective pyrimidylpyrrole inhibitors of extracellular signal-regulated kinase (ERK) using conformational control
利用构象控制进行结构引导设计强效且选择性的胞外信号调节激酶 (ERK) 嘧啶吡咯抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm900630q
Alex M Aronov, Qing Tang, Gabriel Martinez-Botella, Guy W Bemis, Jingrong Cao, Guanjing Chen, Nigel P Ewing, Pamella J Ford, Ursula A Germann, Jeremy Green, Michael R Hale, Marc Jacobs, James W Janetka, Francois Maltais, William Markland, Mark N Namchuk, Suganthini Nanthakumar, Srinivasu Poondru, Ju