日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fluorine-18-Labeled Nucleotide Analogs Targeting Ecto-5'-Nucleotidase (CD73) for Positron Emission Tomography Imaging of Solid Tumors

用于实体瘤正电子发射断层扫描成像的靶向胞外5'-核苷酸酶(CD73)的氟-18标记核苷酸类似物

Dobelmann, Clemens; Schmies, Constanze C; Rolshoven, Georg Wilhelm; Scortichini, Mirko; Wagner, Stefan; Isaak, Andreas; Idris, Riham M; Dabel, Jennifer; Grey, Lucie; Losenkova, Karolina; Moschütz, Susanne; Hroub, Haneen Al; Keim, Antje; Höppner, Sandra; Sandholm, Jouko; Boström, Pia; Hollmén, Maija; Sträter, Norbert; Hermann, Sven; Yegutkin, Gennady G; Jacobson, Kenneth A; Schelhaas, Sonja; Müller, Christa E; Junker, Anna

(N)-Methanocarba Adenosine Derivatives as Dual Modulators of P-Glycoprotein and ABCG2 Transporters

(N)-甲氧基碳腺苷衍生物作为P-糖蛋白和ABCG2转运蛋白的双重调节剂

Murakami, Megumi; Tosh, Dilip K; Salazar, Paula B; Jacobson, Kenneth A; Ambudkar, Suresh V

(N)-Methanocarba-adenosines as monoamine transporter allosteric inhibitors: Extended N(6) groups for bitopic stabilization

(N)-甲氧基碳-腺苷作为单胺转运体变构抑制剂:用于双拓扑稳定的扩展N(6)基团

Tosh, Dilip K; Pavan, Matteo; Kozell, Laura B; Eshleman, Amy J; Schmachtenberg, Jennifer L; Wolfrum, Katherine M; Schutzer, William E; Abbas, Atheir I; Jacobson, Kenneth A

IMMU-82. Neuronal modulation of immunity in glioblastoma

IMMU-82。胶质母细胞瘤中神经元对免疫的调节

Bonifant, Challice L; Shah, Nirali N; Youngblood, Mark; Tripathi, Shashwat; Najem, Hinda; Congivaram, Harrshavasan; Gomez, Mateo; Sears, Thomas; Hurley, Lisa; Billingham, Leah; Silvers, Caylee; Wang, Wenxia; Tiek, Deanna; Sadagopan, Nishanth; Chaliparambil, Rahul; Pu, Qianyi; Wai, Ching Man; Choudhury, Abrar; Steffens, Alicia; McCortney, Kathleen; Cervantes, Gustavo; Oyon, Daniel; Fernandez, Luis; Selner, Ashley; Fares, Jawad; Hagan, Matthew; Trybula, Joy; Yeung, Jacky; Peyre, Matthieu; Kalamarides, Michel; Zhang, Peng; Stegh, Alexander; Ashley, David; Horbinski, Craig; Ahrendsen, Jared; Jamshidi, Pouya; Brat, Daniel; Lukas, Rimas; Stupp, Roger; Lesniak, Maciej; Sonabend, Adam; Dunn, Gavin; Chandler, James; Tate, Matthew; Magill, Stephen; Miska, Jason; Curran, Michael; Raleigh, David; Heimberger, Amy; Du, Ruochen; Hurley, Lisa Agnes; Tripathi, Shashwat; Najem, Hinda; Miska, Jason; Hill, Virginia; Ahrendsen, Jared; Horbinski, Craig; Khatri, Latha; Rao, Ganesh; Waters, Emily Alexandria; Wai, Ching Man; Lukas, Rimas V; Stupp, Roger; Brat, Daniel J; Thorp, Edward B; Lesniak, Maciej S; Heimberger, Amy B; Johnson, Theodore S; Pacholczyk, Rafal; Satpathy, Sarthak; Berrong, Zuzana; Chien, Franklin; Huang, Chenbin; Thomas, Beena E; Chi, Susan N; Baird, Lissa; Sadek, Ramses F; Friedman, Gregory; Hummel, Trent R; Yeo, Kee Kiat; MacDonald, Tobey J; Bhasin, Manoj K; Munn, David H; Hancock, John C; Zhao, Qiuchen; Shaw, Tyler; Seaman, Jonathan; Briceno, Nicole; Pavan, Matteo; Olivia, Paola; Lee, Jihyun; Naylor, Huw; Pitoulias, Matthaios; Pisupati, Venkat; Kishore, Kamal; Porcu, Luca; Mitrophanov, Alexander Y; Natoli, Manuela; Miller, Jodi; Santos, Miguel; Zhang, Meili; Davis, Dionne; Zhang, Wei; Song, Hua; Spurgeon, Jo; Kim, Hye; Hara, Ayaka; Huguely, Caitlin; Anderson, Brita; Steffke, Emily; Keretsu, Seketoulie; Chesler, Alexander T; Yang, Chunzhang; Robinson, Hugh; Jacobson, Kenneth A; Gilbert, Mark R; Terabe, Masaki; Mair, Richard

E. B. Hershberg Award: Taming Inflammation by Tuning Purinergic Signaling

EB Hershberg奖:通过调节嘌呤能信号传导来抑制炎症

Jacobson, Kenneth A

Photoswitchable Diazocine Derivative for Adenosine A(3) Receptor Activation in Psoriasis

用于银屑病腺苷A(3)受体激活的光开关二氮杂辛衍生物

López-Cano, Marc; Scortichini, Mirko; Tosh, Dilip K; Salmaso, Veronica; Ko, Tongil; Salort, Glòria; Filgaira, Ingrid; Soler, Concepció; Trauner, Dirk; Hernando, Jordi; Jacobson, Kenneth A; Ciruela, Francisco

Selective bioorthogonal probe for N-glycan hybrid structures.

用于N-糖杂合结构的选择性生物正交探针

Mukherjee Mana Mohan, Biesbrock Devin, Abramowitz Lara K, Pavan Matteo, Kumar Bhoj, Walter Peter J, Azadi Parastoo, Jacobson Kenneth A, Hanover John A

Abraham Patchornik: The Contemporary Relevance of His Work for Chemistry and Biology

亚伯拉罕·帕乔尼克:他的工作对化学和生物学的当代意义

Jacobson, Kenneth A; Ellis-Davies, Graham C R

Bitopic A(3) Adenosine Receptor Molecular Probes: Positive Allosteric Modulation and Noncanonical Activation

双拓扑A(3)腺苷受体分子探针:正向变构调节和非经典激活

Kurma, Siva Hariprasad; Pavan, Matteo; Wan, Tina C; Pradhan, Balaram; López-Cano, Marc; Ciruela, Francisco; Gao, Zhan-Guo; Auchampach, John A; Jacobson, Kenneth A

UDP-glucose and MRS2905 agonist-bound states of the purinergic P2Y(14) receptor

嘌呤能P2Y(14)受体的UDP-葡萄糖和MRS2905激动剂结合状态

Fay, Jonathan F; Kousouros, Joseph; Gao, Zhan-Guo; Pavan, Matteo; Oliva, Paola; Pramanik, Asmita; Meyer, Clayton; Kurma, Siva Hariprasad; Xu, Wen; Krumm, Brian; Jacobson, Kenneth A