日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MTA-cooperative PRMT5 inhibitors from cofactor-directed DNA-encoded library screens.

通过辅因子导向的DNA编码文库筛选得到的MTA协同PRMT5抑制剂

Andersson Jan, Cowland Sanne, Vestergaard Mikkel, Yang Yajing, Liu Siyuan, Fang Xie, Mukund Susmith, Ghimire-Rijal Sudipa, Carter Chris, Chung Grace, Jacso Tomas, Sarvary Ian, Hughes Paul E, Gouliaev Alex, Payton Marc, Belmontes Brian, Caenepeel Sean, Franch Thomas, Glad Sanne, Husemoen Birgitte, Nielsen Søren Jensby

From DNA-Encoded Library Screening to AM-9747: An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo Efficacy.

从 DNA 编码文库筛选到 AM-9747:一种具有强效口服体内疗效的 MTA 协同 PRMT5 抑制剂

Sarvary Ian, Vestergaard Mikkel, Moretti Loris, Andersson Jan, Peiró Cadahía Jorge, Cowland Sanne, Flagstad Thomas, Franch Thomas, Gouliaev Alex, Husemoen Gitte, Jacso Tomas, Kronborg Titi, Kuropatnicka Aleksandra, Nadali Anna, Madsen Mads, Nielsen So Ren, Pii David, Ryborg So Ren, Soede Camillia, Allen Jennifer R, Bourbeau Matthew, Li Kexue, Liu Qingyian, Lo Mei-Chu, Madoux Franck, Mardirossian Narbe, Moriguchi Jodi, Ngo Rachel, Peng Chi-Chi, Pettus Liping, Tamayo Nuria, Wang Paul, Kapoor Rajiv, Belmontes Brian, Caenepeel Sean, Hughes Paul, Liu Siyuan, Slemmons Katherine K, Yang Yajing, Xie Fang, Ghimire-Rijal Sudipa, Mukund Susmith, Glad Sanne

Parametric Effects of Single Point Incremental Forming on Hardness of AA1100 Aluminium Alloy Sheets

单点渐进成形对AA1100铝合金板材硬度的参数影响

Najm, Sherwan Mohammed; Paniti, Imre; Trzepieciński, Tomasz; Nama, Sami Ali; Viharos, Zsolt János; Jacso, Adam

AMPK and AKT protein kinases hierarchically phosphorylate the N-terminus of the FOXO1 transcription factor, modulating interactions with 14-3-3 proteins

AMPK 和 AKT 蛋白激酶对 FOXO1 转录因子的 N 端进行分级磷酸化,从而调节与 14-3-3 蛋白的相互作用

Maria Saline, Lukas Badertscher, Madita Wolter, Roxanne Lau, Anders Gunnarsson, Tomas Jacso, Tyrrell Norris, Christian Ottmann, Arjan Snijder

Radiation therapy for deep periocular cancer treatments when protons are unavailable: is combining electrons and orthovoltage therapy beneficial?

当质子疗法不可用时,放射疗法对深部眼周癌的治疗有何益处?电子疗法与正电压疗法相结合是否有益?

Martell, Kevin; Poirier, Yannick; Zhang, Tiezhi; Hudson, Alana; Spencer, David; Jacso, Ferenc; Hayashi, Richard; Banerjee, Robyn; Khan, Rao; Wolfe, Nathan; Voroney, Jon-Paul

Assessing the deviation from the inverse square law for orthovoltage beams with closed-ended applicators

评估封闭式施加器正交电压束偏离平方反比定律的情况

Gräfe, James; Poirier, Yannick; Jacso, Ferenc; Khan, Rao; Liu, Hong-Wei; Villarreal-Barajas, J Eduardo

Substrate transport activation is mediated through second periplasmic loop of transmembrane protein MalF in maltose transport complex of Escherichia coli

大肠杆菌麦芽糖转运复合物中跨膜蛋白 MalF 的第二个周质环介导底物转运激活。

Jacso, Tomas; Schneider, Erwin; Rupp, Bernd; Reif, Bernd