日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rational design and in vivo validation of capsid inhibitors for enterovirus D68.

肠道病毒D68衣壳抑制剂的合理设计及体内验证。

Li Kan, Rudy Michael J, Klose Thomas, Tan Haozhou, Wu Xiangmeng, Demssie Hiwot A, Anderson Jacqueline S, Jadhav Prakash, Zhang Qing-Yu, Clarke Penny, Kuhn Richard J, Tyler Kenneth L, Wang Jun

Development of a Fluorescence Polarization Assay for the SARS-CoV-2 Papain-like Protease.

SARS-CoV-2木瓜蛋白酶样蛋白酶的荧光偏振检测方法的开发

Li Kan, Jadhav Prakash, Wen Yu, Tan Haozhou, Wang Jun

Design of a SARS-CoV-2 papain-like protease inhibitor with antiviral efficacy in a mouse model

设计一种在小鼠模型中具有抗病毒功效的SARS-CoV-2木瓜蛋白酶样蛋白酶抑制剂

Tan, Bin; Zhang, Xiaoming; Ansari, Ahmadullah; Jadhav, Prakash; Tan, Haozhou; Li, Kan; Chopra, Ashima; Ford, Alexandra; Chi, Xiang; Ruiz, Francesc Xavier; Arnold, Eddy; Deng, Xufang; Wang, Jun

Structure-Based Design of Covalent SARS-CoV-2 Papain-like Protease Inhibitors.

基于结构的共价SARS-CoV-2木瓜蛋白酶样蛋白酶抑制剂设计

Tan Bin, Liang Xueying, Ansari Ahmadullah, Jadhav Prakash, Tan Haozhou, Li Kan, Ruiz Francesc Xavier, Arnold Eddy, Deng Xufang, Wang Jun

Structure-Based Lead Optimization of Enterovirus D68 2A Protease Inhibitors

基于结构的肠道病毒D68 2A蛋白酶抑制剂先导化合物优化

Tan, Bin; Liu, Chang; Li, Kan; Jadhav, Prakash; Lambrinidis, George; Zhu, Lan; Olson, Linda; Tan, Haozhou; Wen, Yu; Kolocouris, Antonios; Liu, Wei; Wang, Jun

Design of SARS-CoV-2 papain-like protease inhibitor with antiviral efficacy in a mouse model

设计一种在小鼠模型中具有抗病毒功效的SARS-CoV-2木瓜蛋白酶样蛋白酶抑制剂

Tan, Bin; Zhang, Xiaoming; Ansari, Ahmadullah; Jadhav, Prakash; Tan, Haozhou; Li, Kan; Chopra, Ashima; Ford, Alexandra; Chi, Xiang; Ruiz, Francesc Xavier; Arnold, Eddy; Deng, Xufang; Wang, Jun

Progress and Challenges in Targeting the SARS-CoV-2 Papain-like Protease

针对SARS-CoV-2木瓜蛋白酶样蛋白酶的研究进展与挑战

Tan, Haozhou; Hu, Yanmei; Jadhav, Prakash; Tan, Bin; Wang, Jun

Gold-catalyzed (4 + 2)-annulations between α-alkyl alkenylgold carbenes and benzisoxazoles with reactive alkyl groups

金催化的α-烷基烯基金卡宾与具有活性烷基的苯并异噁唑之间的(4+2)环加成反应

Mokar, Bhanudas Dattatray; Jadhav, Prakash D; Pandit, Y B; Liu, Rai-Shung

Total Syntheses and Biological Evaluation of (±)-Botryosphaeridione, (±)-Pleodendione, 4-epi-Periconianone B, and Analogues

(±)-Botryosphaeridione、(±)-Pleodendione、4-epi-Periconianone B 及其类似物的全合成和生物学评价

Handore, Kishor L; Jadhav, Prakash D; Hazra, Bibhabasu; Basu, Anirban; Reddy, D Srinivasa