日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
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2025
2026
影响因子:
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Population pharmacokinetic and pharmacokinetic-pharmacodynamic modeling of bempedoic acid and low-density lipoprotein cholesterol in healthy subjects and patients with dyslipidemia

在健康受试者和血脂异常患者中，贝培多酸和低密度脂蛋白胆固醇的群体药代动力学和药代动力学-药效学模型

期刊:Journal of Pharmacokinetics and Pharmacodynamics
影响因子:2.8
doi:10.1007/s10928-023-09864-w
Jadhav, Satyawan B; Amore, Benny M; Bockbrader, Howard; Crass, Ryan L; Chapel, Sunny; Sasiela, William J; Emery, Maurice G
心血管
代谢
发表日期：2023
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Pharmacodynamic effect of bempedoic acid and statin combinations: predictions from a dose-response model

贝培多酸与他汀类药物联合用药的药效学效应：基于剂量反应模型的预测

期刊:European Heart Journal-Cardiovascular Pharmacotherapy
影响因子:6.1
doi:10.1093/ehjcvp/pvab064
Jadhav, Satyawan B; Crass, Ryan L; Chapel, Sunny; Kerschnitzki, Michael; Sasiela, William J; Emery, Maurice G; Amore, Benny M; Barrett, P Hugh R; Watts, Gerald F; Catapano, Alberico L
发表日期：2022
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Tetrahydronaphthyridine and dihydronaphthyridinone ethers as positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu₠).

四氢萘啶和二氢萘啶酮醚作为代谢型谷氨酸受体 5 (mGluâ‚) 的正向变构调节剂

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm500259z
Turlington Mark, Malosh Chrysa, Jacobs Jon, Manka Jason T, Noetzel Meredith J, Vinson Paige N, Jadhav Satyawan, Herman Elizabeth J, Lavreysen Hilde, Mackie Claire, Bartolomé-Nebreda José M, Conde-Ceide Susana, Martín-Martín M Luz, Tong Han Min, López Silvia, MacDonald Gregor J, Steckler Thomas, Daniels J Scott, Weaver C David, Niswender Colleen M, Jones Carrie K, Conn P Jeffrey, Lindsley Craig W, Stauffer Shaun R
代谢
发表日期：2014
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Dihydrothiazolopyridone derivatives as a novel family of positive allosteric modulators of the metabotropic glutamate 5 (mGlu5) receptor.

二氢噻唑并吡啶酮衍生物作为代谢型谷氨酸 5 (mGlu5) 受体的一类新型正向变构调节剂

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm400650w
Bartolomé-Nebreda José Manuel, Conde-Ceide Susana, Delgado Francisca, Iturrino Laura, Pastor Joaquín, Pena Miguel Ángel, Trabanco Andrés A, Tresadern Gary, Wassvik Carola M, Stauffer Shaun R, Jadhav Satyawan, Gogi Kiran, Vinson Paige N, Noetzel Meredith J, Days Emily, Weaver C David, Lindsley Craig W, Niswender Colleen M, Jones Carrie K, Conn P Jeffrey, Rombouts Frederik, Lavreysen Hilde, Macdonald Gregor J, Mackie Claire, Steckler Thomas
代谢
发表日期：2013
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3-Cyano-5-fluoro-N-arylbenzamides as negative allosteric modulators of mGlu(5): Identification of easily prepared tool compounds with CNS exposure in rats

3-氰基-5-氟-N-芳基苯甲酰胺作为mGlu(5)的负变构调节剂：易于制备的工具化合物在大鼠中枢神经系统暴露中的鉴定

期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2010.06.064
Felts, Andrew S; Lindsley, Stacey R; Lamb, Jeffrey P; Rodriguez, Alice L; Menon, Usha N; Jadhav, Satyawan; Jones, Carrie K; Conn, P Jeffrey; Lindsley, Craig W; Emmitte, Kyle A
Rat
神经科学
发表日期：2010
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