日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Plasmodiumfalciparum protein kinase 6 and hemozoin formation are inhibited by a type II human kinase inhibitor exhibiting antimalarial activity

一种具有抗疟活性的II型人激酶抑制剂可抑制恶性疟原虫蛋白激酶6和血红素的形成。

Flore Nardella ,Tiantian Jiang ,Lushun Wang ,Monica J Bohmer ,Subhoja Chakraborty ,John Okombo ,Jaeson Calla ,Tatiane Macedo Silva ,Samuel Pazicky ,Jianwei Che ,Jin Jeon ,Evie Vincent ,Nonlawat Boonyalai ,Rachael Coyle ,Mairi J Buchanan ,Samuel Schaefer ,Daisy Chen ,Amaan Khan ,Emily Mayville ,Mariana Laureano De Souza ,Mayland Treat ,Jordan Charlton ,Patrick K Tumwebaze ,Seth Tjia ,Lukas Montejo ,Karen Cover ,Philip J Rosenthal ,Roland A Cooper ,Zbynek Bozdech ,Marcus C S Lee ,Ratna Chakrabarti ,Sanjay A Desai ,David A Fidock ,Jinhua Wang ,Nathanael S Gray ,Elizabeth A Winzeler ,Debopam Chakrabarti

Human nuclear hormone receptor activity contributes to malaria parasite liver stage development

人类核激素受体活性促进疟原虫肝脏阶段的发展

Nimisha Mittal, Chadwick Davis, Peter McLean, Jaeson Calla, Karla P Godinez-Macias, Alison Gardner, David Healey, Pamela Orjuela-Sanchez, Sabine Ottilie, Yolanda Chong, Christopher Gibson, Elizabeth A Winzeler

Development of Potent and Highly Selective Epoxyketone-Based Plasmodium Proteasome Inhibitors

开发强效、高选择性的基于环氧酮的疟原虫蛋白酶体抑制剂

Jehad Almaliti, Pavla Fajtová, Jaeson Calla, Gregory M LaMonte, Mudong Feng, Frances Rocamora, Sabine Ottilie, Evgenia Glukhov, Evzen Boura, Raymond T Suhandynata, Jeremiah D Momper, Michael K Gilson, Elizabeth A Winzeler, William H Gerwick, Anthony J O'Donoghue

A novel CSP C-terminal epitope targeted by an antibody with protective activity against Plasmodium falciparum

一种具有抗恶性疟原虫保护活性的抗体靶向的新型 CSP C 端表位

Nathan Beutler, Tossapol Pholcharee, David Oyen, Yevel Flores-Garcia, Randall S MacGill, Elijah Garcia, Jaeson Calla, Mara Parren, Linlin Yang, Wayne Volkmuth, Emily Locke, Jason A Regules, Sheetij Dutta, Daniel Emerling, Angela M Early, Daniel E Neafsey, Elizabeth A Winzeler, C Richter King, Fidel

Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials

探索开放全球健康化学多样性库,寻找下一代抗疟药物的多阶段活性起点

Matthew Abraham, Kerstin Gagaring, Marisa L Martino, Manu Vanaerschot, David M Plouffe, Jaeson Calla, Karla P Godinez-Macias, Alan Y Du, Melanie Wree, Yevgeniya Antonova-Koch, Korina Eribez, Madeline R Luth, Sabine Ottilie, David A Fidock, Case W McNamara, Elizabeth A Winzeler

Dual RNA-seq identifies human mucosal immunity protein Mucin-13 as a hallmark of Plasmodium exoerythrocytic infection

双 RNA 测序鉴定出人类粘膜免疫蛋白 Mucin-13 是疟原虫红细胞外感染的标志

Gregory M LaMonte, Pamela Orjuela-Sanchez, Jaeson Calla, Lawrence T Wang, Shangzhong Li, Justine Swann, Annie N Cowell, Bing Yu Zou, Alyaa M Abdel-Haleem Mohamed, Zaira Hellen Villa Galarce, Marta Moreno, Carlos Tong Rios, Joseph M Vinetz, Nathan Lewis, Elizabeth A Winzeler