日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Activation of CB2R by synthetic CB2R agonist, PM289, improves brain endothelial barrier properties, decreases inflammatory response and enhances endothelial repair

合成 CB2R 激动剂 PM289 激活 CB2R,可改善脑内皮屏障特性、降低炎症反应并增强内皮修复

Trent A Bullock, Kalpani N Udeni Galpayage Dona, Jonathan F Hale, Paula Morales, Nadine Jagerovic, Allison M Andrews, Servio H Ramirez

Administration of Linoleoylethanolamide Reduced Weight Gain, Dyslipidemia, and Inflammation Associated with High-Fat-Diet-Induced Obesity

服用亚油酰乙醇酰胺可减少高脂饮食引起的肥胖相关的体重增加、血脂异常和炎症

Rubén Tovar, Marialuisa de Ceglia, Massimo Ubaldi, Miguel Rodríguez-Pozo, Laura Soverchia, Carlo Cifani, Gema Rojo, Ana Gavito, Laura Hernandez-Folgado, Nadine Jagerovic, Roberto Ciccocioppo, Elena Baixeras, Fernando Rodríguez de Fonseca, Juan Decara

The Binding Mode to Orthosteric Sites and/or Exosites Underlies the Therapeutic Potential of Drugs Targeting Cannabinoid CB(2) Receptors

靶向大麻素 CB(2) 受体的药物的治疗潜力取决于其与正构位点和/或外位点的结合模式。

Franco, Rafael; Morales, Paula; Navarro, Gemma; Jagerovic, Nadine; Reyes-Resina, Irene

Palmitoleoylethanolamide Is an Efficient Anti-Obesity Endogenous Compound: Comparison with Oleylethanolamide in Diet-Induced Obesity

棕榈油酰乙醇酰胺是一种有效的抗肥胖内源性化合物:与饮食引起的肥胖中的油酰乙醇酰胺进行比较

Rubén Tovar, Ana Luisa Gavito, Antonio Vargas, Laura Soverchia, Laura Hernandez-Folgado, Nadine Jagerovic, Elena Baixeras, Roberto Ciccocioppo, Fernando Rodríguez de Fonseca, Juan Decara

Preclinical Investigation in Neuroprotective Effects of the GPR55 Ligand VCE-006.1 in Experimental Models of Parkinson's Disease and Amyotrophic Lateral Sclerosis

GPR55 配体 VCE-006.1 对帕金森病和肌萎缩侧索硬化症实验模型的神经保护作用的临床前研究

Sonia Burgaz, Concepción García, Claudia Gonzalo-Consuegra, Marta Gómez-Almería, Francisco Ruiz-Pino, Juan Diego Unciti, María Gómez-Cañas, Juan Alcalde, Paula Morales, Nadine Jagerovic, Carmen Rodríguez-Cueto, Eva de Lago, Eduardo Muñoz, Javier Fernández-Ruiz

Discovery of Homobivalent Bitopic Ligands of the Cannabinoid CB(2) Receptor*

大麻素CB(2)受体同源二价双位配体的发现*

Morales, Paula; Navarro, Gemma; Gómez-Autet, Marc; Redondo, Laura; Fernández-Ruiz, Javier; Pérez-Benito, Laura; Cordomí, Arnau; Pardo, Leonardo; Franco, Rafael; Jagerovic, Nadine

Antitumor Cannabinoid Chemotypes: Structural Insights

抗肿瘤大麻素化学类型:结构见解

Morales, Paula; Jagerovic, Nadine

Chromenopyrazole, a Versatile Cannabinoid Scaffold with in Vivo Activity in a Model of Multiple Sclerosis

色诺吡唑是一种多功能大麻素支架,在多发性硬化症模型中具有体内活性

Paula Morales, María Gómez-Cañas #, Gemma Navarro #, Dow P Hurst, Francisco J Carrillo-Salinas, Laura Lagartera, Ruth Pazos, Pilar Goya, Patricia H Reggio, Carmen Guaza, Rafael Franco, Javier Fernández-Ruiz, Nadine Jagerovic

Targeting Cannabinoid CB2 Receptors in the Central Nervous System. Medicinal Chemistry Approaches with Focus on Neurodegenerative Disorders

靶向中枢神经系统中的大麻素CB2受体:以神经退行性疾病为重点的药物化学方法

Navarro, Gemma; Morales, Paula; Rodríguez-Cueto, Carmen; Fernández-Ruiz, Javier; Jagerovic, Nadine; Franco, Rafael

Benzyl-1,2,4-triazoles as CB 1 Cannabinoid Receptor Ligands: Preparation and In Vitro Pharmacological Evaluation

苄基-1,2,4-三唑类化合物作为CB1大麻素受体配体:制备及体外药理学评价

Hernandez-Folgado, Laura; Decara, Juan; Rodríguez de Fonseca, Fernando; Goya, Pilar; Jagerovic, Nadine