Allosteric modulation of AURKA kinase activity by a small-molecule inhibitor of its protein-protein interaction with TPX2
通过小分子抑制剂对 AURKA 激酶活性进行变构调节,抑制其与 TPX2 的蛋白质-蛋白质相互作用
期刊:Scientific Reports
影响因子:3.8
doi:10.1038/srep28528
Matej Janeček, Maxim Rossmann, Pooja Sharma, Amy Emery, David J Huggins, Simon R Stockwell, Jamie E Stokes, Yaw S Tan, Estrella Guarino Almeida, Bryn Hardwick, Ana J Narvaez, Marko Hyvönen, David R Spring, Grahame J McKenzie, Ashok R Venkitaraman