日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ReCHEMbinant stapling enhances intracellular delivery and bioactivity of engineered protein inhibitors

ReCHEMbinant 交联技术可增强工程化蛋白抑制剂的细胞内递送和生物活性。

Kahler, Jan Pascal; Ellenbroek, Brecht D; van der Noord, Vera E; van de Water, Bob; Pomplun, Sebastian J

Development of DuoMYC: a synthetic cell penetrant miniprotein that efficiently inhibits the oncogenic transcription factor MYC

DuoMYC的研发:一种能有效抑制致癌转录因子MYC的合成细胞穿透性小蛋白

Ellenbroek, Brecht D; Kahler, Jan Pascal; Arella, Damiano; Lin, Cherina; Jespers, Willem; Züger, Eliane Ann-Katrin; Drukker, Micha; Pomplun, Sebastian J

Duodenal macrophages control dietary iron absorption via local degradation of transferrin

十二指肠巨噬细胞通过局部降解转铁蛋白来控制膳食铁的吸收。

Sukhbaatar, Nyamdelger; Schöller, Maria; Fritsch, Stephanie Deborah; Linke, Monika; Horer, Stefanie; Träger, Manuela; Mazić, Mario; Forisch, Stephan; Gonzales, Karine; Kahler, Jan Pascal; Binder, Carina; Lassnig, Caroline; Strobl, Birgit; Müller, Mathias; Scheiber-Mojdehkar, Barbara; Gundacker, Claudia; Dabsch, Stefanie; Kain, Renate; Hengstschläger, Markus; Verhelst, Steven H L; Weiss, Günter; Theurl, Igor; Weichhart, Thomas

Phosphinate esters as novel warheads for activity-based probes targeting serine proteases

膦酸酯作为新型活性探针,靶向丝氨酸蛋白酶

Kahler, Jan Pascal; Verhelst, Steven H L

ATP13A2 deficiency disrupts lysosomal polyamine export

ATP13A2 缺乏会破坏溶酶体多胺输出

Sarah van Veen #, Shaun Martin #, Chris Van den Haute, Veronick Benoy, Joseph Lyons, Roeland Vanhoutte, Jan Pascal Kahler, Jean-Paul Decuypere, Géraldine Gelders, Eric Lambie, Jeffrey Zielich, Johannes V Swinnen, Wim Annaert, Patrizia Agostinis, Bart Ghesquière, Steven Verhelst, Veerle Baekelandt, J

Facile Synthesis of Aminomethyl Phosphinate Esters as Serine Protease Inhibitors with Primed Site Interaction

简便合成氨甲基膦酸酯类化合物作为丝氨酸蛋白酶抑制剂及其与起始位点的相互作用

Kahler, Jan Pascal; Lenders, Stijn; van de Plassche, Merel A T; Verhelst, Steven H L

Cellular metabolism constrains innate immune responses in early human ontogeny

细胞代谢限制了人类早期个体发育过程中的先天免疫反应

Bernard Kan,Christina Michalski,Helen Fu,Hilda H T Au,Kelsey Lee,Elizabeth A Marchant,Maye F Cheng,Emily Anderson-Baucum,Michal Aharoni-Simon,Peter Tilley,Raghavendra G Mirmira,Colin J Ross,Dan S Luciani,Eric Jan,Pascal M Lavoie

Cellular metabolism constrains innate immune responses in early human ontogeny

细胞代谢限制了人类早期个体发育过程中的先天免疫反应

Bernard Kan ,Christina Michalski ,Helen Fu ,Hilda H T Au ,Kelsey Lee ,Elizabeth A Marchant ,Maye F Cheng ,Emily Anderson-Baucum ,Michal Aharoni-Simon ,Peter Tilley ,Raghavendra G Mirmira ,Colin J Ross ,Dan S Luciani ,Eric Jan ,Pascal M Lavoie