A positive allosteric modulator of the β1AR with antagonist activity for catecholaminergic polymorphic ventricular tachycardia
β1AR 的正向变构调节剂,对儿茶酚胺能多形性室性心动过速具有拮抗活性
期刊:Journal of Clinical Investigation
影响因子:13.3
doi:10.1172/JCI190252.
Alyssa Grogan ,Robin M Perelli ,Seungkirl Ahn ,Haoran Jiang ,Arun Jyothidasan ,Damini Sood ,Chongzhao You ,David I Israel ,Alex Shaginian ,Qiuxia Chen ,Jian Liu ,Jialu Wang ,Jan Steyaert ,Alem W Kahsai ,Andrew P Landstrom ,Robert J Lefkowitz ,Howard A Rockman