日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A positive allosteric modulator of the β1AR with antagonist activity for catecholaminergic polymorphic ventricular tachycardia

β1AR 的正向变构调节剂,对儿茶酚胺能多形性室性心动过速具有拮抗活性

Alyssa Grogan ,Robin M Perelli ,Seungkirl Ahn ,Haoran Jiang ,Arun Jyothidasan ,Damini Sood ,Chongzhao You ,David I Israel ,Alex Shaginian ,Qiuxia Chen ,Jian Liu ,Jialu Wang ,Jan Steyaert ,Alem W Kahsai ,Andrew P Landstrom ,Robert J Lefkowitz ,Howard A Rockman

Structural basis of antimicrobial membrane coat assembly by human GBP1

人类GBP1组装抗菌膜涂层的结构基础

Tanja Kuhm, Clémence Taisne, Cecilia de Agrela Pinto, Luca Gross, Evdokia A Giannopoulou, Stefan T Huber, Els Pardon, Jan Steyaert, Sander J Tans, Arjen J Jakobi

Investigating the In Vivo Effects of Anti-Prion Protein Nanobodies on Prion Disease with AAV Vector

利用AAV载体研究抗朊病毒蛋白纳米抗体对朊病毒疾病的体内作用

Jingjing Zhang ,Mengfei Wang ,Dan Wang ,Xiangyi Zhang ,Yue Ma ,Els Pardon ,Jan Steyaert ,Romany Abskharon ,Fei Wang ,Jiyan Ma

Structural insights into Frizzled3 through nanobody modulators

通过纳米抗体调节剂深入了解 Frizzled3 的结构

James Hillier #, Yuguang Zhao #, Loic Carrique, Tomas Malinauskas, Reinis R Ruza, Tao-Hsin Chang, Gangshun Yi, Helen M E Duyvesteyn, Jing Yu, Weixian Lu, Els Pardon, Jan Steyaert, Yanan Zhu, Tao Ni, E Yvonne Jones

Structural basis of μ-opioid receptor targeting by a nanobody antagonist

纳米抗体拮抗剂靶向μ-阿片受体的结构基础

Jun Yu #,Amit Kumar #,Xuefeng Zhang,Charlotte Martin,Kevin Van Holsbeeck,Pierre Raia,Antoine Koehl,Toon Laeremans,Jan Steyaert,Aashish Manglik,Steven Ballet,Andreas Boland,Miriam Stoeber

Structural basis of thiamine transport and drug recognition by SLC19A3

SLC19A3 硫胺素转运和药物识别的结构基础

Florian Gabriel, Lea Spriestersbach, Antonia Fuhrmann, Katharina E J Jungnickel, Siavash Mostafavi, Els Pardon, Jan Steyaert, Christian Löw

Crystal structure of human serum albumin in complex with megabody reveals unique human and murine cross-reactive binding site

人血清白蛋白与巨抗体复合物的晶体结构揭示了独特的人类和鼠交叉反应结合位点

Sofia De Felice, Zhanna Romanyuk, Monica Chinellato, Giulia Zoia, Sara Linciano, Yoichi Kumada, Els Pardon, Jan Steyaert, Alessandro Angelini, Laura Cendron

Structural basis for the allosteric modulation of rhodopsin by nanobody binding to its extracellular domain

纳米抗体与视紫红质胞外结构域结合对其变构调节的结构基础

Arum Wu #, David Salom #, John D Hong, Aleksander Tworak, Kohei Watanabe, Els Pardon, Jan Steyaert, Hideki Kandori, Kota Katayama, Philip D Kiser, Krzysztof Palczewski

Structural basis of purine nucleotide inhibition of human uncoupling protein 1

嘌呤核苷酸抑制人类解偶联蛋白1的结构基础

Scott A Jones, Prerana Gogoi, Jonathan J Ruprecht, Martin S King, Yang Lee, Thomas Zögg, Els Pardon, Deepak Chand, Stefan Steimle, Danielle M Copeman, Camila A Cotrim, Jan Steyaert, Paul G Crichton, Vera Moiseenkova-Bell, Edmund R S Kunji

Structural Basis of μ-Opioid Receptor-Targeting by a Nanobody Antagonist

纳米抗体拮抗剂靶向 μ-阿片受体的结构基础

Jun Yu, Amit Kumar, Xuefeng Zhang, Charlotte Martin, Pierre Raia, Antoine Koehl, Toon Laeremans, Jan Steyaert, Aashish Manglik, Steven Ballet, Andreas Boland, Miriam Stoeber