日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Recurrent Resistance Mutations to Lirafugratinib Inform Treatment Sequencing in FGFR2-Driven Tumors.

对利拉夫格拉替尼的复发性耐药突变可指导 FGFR2 驱动肿瘤的治疗顺序。

Facchinetti Francesco, Hollebecque Antoine, Barbé Rémy, Jang Dong Man, Alonso-De-Castro Beatriz, Brayé Floriane, Bigot Ludovic, Nobre Catline, Da Silva Alice, Méteau Mélissandre, Delavigne Mathis, Soares Miguel, Italiano Antoine, Rodriguez Julieta, Mosele Fernanda, Beshiri Kristi, Ducreux Michel, Boilève Alice, Nikolaev Sergey, Alonso-Garcia Inmaculada, Vasseur Damien, Smolenschi Cristina, Bourien Héloise, Cotteret Sophie, Samaniego Juliette, Bernard Elsa, Nicotra Claudio, Ngo-Camus Maud, Nakazawa Seshiru, Tselikas Lambros, Badoual Cécile, André Fabrice, Eck Michael J, Olaussen Ken A, Loriot Yohann, Friboulet Luc

Structural insights into SetA-mediated Rab1 glucosylation and PI3P-guided localization during early Legionella infection

早期军团菌感染过程中SetA介导的Rab1糖基化和PI3P引导的定位的结构解析

Im, Ha Na; Lee, Yeon; Song, Yunju; Hahn, Hyunggu; Jeon, Hyerry; Shin, Donghyuk; Lee, Sangho; Kim, Kyung-Hee; Kim, Kyung-Tae; Suh, Se Won; Jang, Dong Man; Kim, Hyoun Sook

Cryo-EM structures of CRAF/MEK1/14-3-3 complexes in autoinhibited and open-monomer states reveal features of RAF regulation.

CRAF/MEK1/14-3-3 复合物在自身抑制和开放单体状态下的冷冻电镜结构揭示了 RAF 调控的特征

Jang Dong Man, Boxer Kayla, Ha Byung Hak, Tkacik Emre, Levitz Talya, Rawson Shaun, Metivier Rebecca J, Schmoker Anna, Jeon Hyesung, Eck Michael J

Characterization and inhibitor sensitivity of ARAF, BRAF, and CRAF kinases

ARAF、BRAF 和 CRAF 激酶的特性及抑制剂敏感性

Tkacik, Emre; Jang, Dong Man; Boxer, Kayla; Ha, Byung Hak; Eck, Michael J

RAF isoform selectivity of MEK inhibitors and rational design of a covalent ARAF-MEK inhibitor

MEK抑制剂的RAF亚型选择性及共价ARAF-MEK抑制剂的合理设计

Chakraborty, Sayan; Jiang, Jie; Camallonga, Javier Vinals; Gazgalis, Dimitris; Gero, Thomas W; Tavares, Maurício T; Dittemore, Georgia; Tkacik, Emre; Jang, Dong Man; Ha, Byung Hak; Gottlieb, Felix H; Levitz, Talya; Metivier, Rebecca J; Schmoker, Anna M; Scott, David A; Jeon, Hyesung; Jänne, Pasi A; Eck, Michael J

Structural Basis of Inhibition of DCLK1 by Ruxolitinib

鲁索替尼抑制DCLK1的结构基础

Jang, Dong Man; Lim, Hyo Jin; Hahn, Hyunggu; Lee, Yeon; Kim, Hark Kyun; Kim, Hyoun Sook

Family-based exome sequencing combined with linkage analyses identifies rare susceptibility variants of MUC4 for gastric cancer

基于家族的外显子组测序结合连锁分析,鉴定出MUC4基因的罕见易感变异,这些变异与胃癌相关。

Choi, Yoon Jin; Ohn, Jung Hun; Kim, Nayoung; Kim, Wonji; Park, Kyungtaek; Won, Sungho; Sael, Lee; Shin, Cheol Min; Lee, Sun Min; Lee, Sejoon; An, Hyun Joo; Jang, Dong Man; Han, Byung Woo; Lee, Hye Seung; Kang, Seung Joo; Kim, Joo Sung; Lee, Dong Ho