日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cryo-EM structure determination of small therapeutic protein targets at 3 Å-resolution using a rigid imaging scaffold

使用刚性成像支架以 3 Å 分辨率测定小型治疗性蛋白质靶点的低温电子显微镜结构

Roger Castells-Graells, Kyle Meador, Mark A Arbing, Michael R Sawaya, Morgan Gee, Duilio Cascio, Emma Gleave, Judit É Debreczeni, Jason Breed, Karoline Leopold, Ankoor Patel, Dushyant Jahagirdar, Bronwyn Lyons, Sriram Subramaniam, Chris Phillips, Todd O Yeates

KRAS-specific inhibition using a DARPin binding to a site in the allosteric lobe

使用 DARPin 与变构叶中的位点结合来进行 KRAS 特异性抑制

Nicolas Bery, Sandrine Legg, Judit Debreczeni, Jason Breed, Kevin Embrey, Christopher Stubbs, Paulina Kolasinska-Zwierz, Nathalie Barrett, Rose Marwood, Jo Watson, Jon Tart, Ross Overman, Ami Miller, Christopher Phillips, Ralph Minter, Terence H Rabbitts

Structural and functional characterization of a DARPin which inhibits Ras nucleotide exchange

抑制 Ras 核苷酸交换的 DARPin 的结构和功能表征

Sandrine Guillard, Paulina Kolasinska-Zwierz, Judit Debreczeni, Jason Breed, Jing Zhang, Nicolas Bery, Rose Marwood, Jon Tart, Ross Overman, Pawel Stocki, Bina Mistry, Christopher Phillips, Terence Rabbitts, Ronald Jackson, Ralph Minter

MTH1 Substrate Recognition--An Example of Specific Promiscuity

MTH1 底物识别——特定混杂性的一个例子

J Willem M Nissink, Michal Bista, Jason Breed, Nikki Carter, Kevin Embrey, Jonathan Read, Jon J Winter-Holt

Discovery of cofactor-specific, bactericidal Mycobacterium tuberculosis InhA inhibitors using DNA-encoded library technology

利用 DNA 编码库技术发现辅助因子特异性、杀菌性结核分枝杆菌 InhA 抑制剂

Holly H Soutter, Paolo Centrella, Matthew A Clark, John W Cuozzo, Christoph E Dumelin, Marie-Aude Guie, Sevan Habeshian, Anthony D Keefe, Kaitlyn M Kennedy, Eric A Sigel, Dawn M Troast, Ying Zhang, Andrew D Ferguson, Gareth Davies, Eleanor R Stead, Jason Breed, Prashanti Madhavapeddi, Jon A Read3