日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Novel, Long-Acting, Small Molecule PKM2 Activator and Its Potential Broad Application Against Photoreceptor Degeneration

一种新型长效小分子PKM2激活剂及其在对抗光感受器退行性疾病方面的潜在广泛应用

Warren W Pan,Katherine M Weh,Sraboni Chaudhury,Roshini Fernando,Heather Hager,Bo Wen,Krishnapriya Chinnaswamy,Jeanne A Stuckey ,Jason C Rech,Cagri G Besirli,Eric Weh,Thomas J Wubben

Prophylactic Mitigation of Acute Graft versus Host Disease by Novel 2-(Pyrrolidin-1-ylmethyl)pyrrole-Based Stimulation-2 (ST2) Inhibitors

新型 2-(吡咯烷-1-基甲基)吡咯基刺激-2 (ST2) 抑制剂预防性缓解急性移植物抗宿主病

Xinrui Yuan, Hua Jiang, Denggang Fu, Jason C Rech, Aaron Robida, Krishani Rajanayake, Hebao Yuan, Miao He, Bo Wen, Duxin Sun, Chen Liu, Krishnapriya Chinnaswamy, Jeanne A Stuckey, Sophie Paczesny, Chao-Yie Yang

Development of Novel Small-Molecule Activators of Pyruvate Kinase Muscle Isozyme 2, PKM2, to Reduce Photoreceptor Apoptosis

开发新型丙酮酸激酶肌肉同工酶 2(PKM2)小分子激活剂以减少感光细胞凋亡

Thomas J Wubben, Sraboni Chaudhury, Brennan T Watch, Jeanne A Stuckey, Eric Weh, Roshini Fernando, Moloy Goswami, Mercy Pawar, Jason C Rech, Cagri G Besirli

From proteomics to discovery of first-in-class ST2 inhibitors active in vivo

从蛋白质组学到发现首创的体内活性 ST2 抑制剂

Abdulraouf M Ramadan, Etienne Daguindau, Jason C Rech, Krishnapriya Chinnaswamy, Jilu Zhang, Greg L Hura, Brad Griesenauer, Zachary Bolten, Aaron Robida, Martha Larsen, Jeanne A Stuckey, Chao-Yie Yang, Sophie Paczesny