日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemical systems biology reveals mechanisms of glucocorticoid receptor signaling

化学系统生物学揭示糖皮质激素受体信号传导机制

Nelson E Bruno ,Jerome C Nwachukwu ,Sathish Srinivasan ,Charles C Nettles ,Tina Izard ,Zhuang Jin ,Jason Nowak ,Michael D Cameron ,Siddaraju V Boregowda ,Donald G Phinney ,Olivier Elemento ,Xu Liu ,Eric A Ortlund ,René Houtman ,Diana A Stavreva ,Gordon L Hager ,Theodore M Kamenecka ,Douglas J Kojetin ,Kendall W Nettles

Didehydro-Cortistatin A Inhibits HIV-1 by Specifically Binding to the Unstructured Basic Region of Tat

二脱氢皮质抑素 A 通过特异性结合 Tat 的非结构化碱性区域来抑制 HIV-1

Sonia Mediouni, Krishna Chinthalapudi, Mary K Ekka, Ippei Usui, Joseph A Jablonski, Mark A Clementz, Guillaume Mousseau, Jason Nowak, Venkat R Macherla, Jacob N Beverage, Eduardo Esquenazi, Phil Baran, Ian Mitchelle S de Vera, Douglas Kojetin, Erwann P Loret, Kendall Nettles, Souvik Maiti, Tina Izar

The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells

SERM/SERD 巴曲昔芬破坏 ESR1 螺旋 12,以克服乳腺癌细胞获得性激素耐药性

Sean W Fanning, Rinath Jeselsohn, Venkatasubramanian Dharmarajan, Christopher G Mayne, Mostafa Karimi, Gilles Buchwalter, René Houtman, Weiyi Toy, Colin E Fowler, Ross Han, Muriel Lainé, Kathryn E Carlson, Teresa A Martin, Jason Nowak, Jerome C Nwachukwu, David J Hosfield, Sarat Chandarlapaty, Emad

Structural and Molecular Mechanisms of Cytokine-Mediated Endocrine Resistance in Human Breast Cancer Cells

人类乳腺癌细胞中细胞因子介导的内分泌抗性的结构和分子机制

Joshua D Stender, Jerome C Nwachukwu, Irida Kastrati, Yohan Kim, Tobias Strid, Maayan Yakir, Sathish Srinivasan, Jason Nowak, Tina Izard, Erumbi S Rangarajan, Kathryn E Carlson, John A Katzenellenbogen, Xin-Qiu Yao, Barry J Grant, Hon S Leong, Chin-Yo Lin, Jonna Frasor, Kendall W Nettles, Christophe

Full antagonism of the estrogen receptor without a prototypical ligand side chain

无需原型配体侧链即可完全拮抗雌激素受体

Sathish Srinivasan, Jerome C Nwachukwu, Nelson E Bruno, Venkatasubramanian Dharmarajan, Devrishi Goswami, Irida Kastrati, Scott Novick, Jason Nowak, Valerie Cavett, Hai-Bing Zhou, Nittaya Boonmuen, Yuechao Zhao, Jian Min, Jonna Frasor, Benita S Katzenellenbogen, Patrick R Griffin, John A Katzenellen

Structural mechanism for signal transduction in RXR nuclear receptor heterodimers

RXR 核受体异二聚体信号转导的结构机制

Douglas J Kojetin, Edna Matta-Camacho, Travis S Hughes, Sathish Srinivasan, Jerome C Nwachukwu, Valerie Cavett, Jason Nowak, Michael J Chalmers, David P Marciano, Theodore M Kamenecka, Andrew I Shulman, Mark Rance, Patrick R Griffin, John B Bruning, Kendall W Nettles

Resveratrol modulates the inflammatory response via an estrogen receptor-signal integration network

白藜芦醇通过雌激素受体信号整合网络调节炎症反应

Jerome C Nwachukwu, Sathish Srinivasan, Nelson E Bruno, Alexander A Parent, Travis S Hughes, Julie A Pollock, Olsi Gjyshi, Valerie Cavett, Jason Nowak, Ruben D Garcia-Ordonez, René Houtman, Patrick R Griffin, Douglas J Kojetin, John A Katzenellenbogen, Michael D Conkright, Kendall W Nettles

Ligand-binding dynamics rewire cellular signaling via estrogen receptor-α

配体结合动力学通过雌激素受体-α 重新连接细胞信号传导

Sathish Srinivasan, Jerome C Nwachukwu, Alex A Parent, Valerie Cavett, Jason Nowak, Travis S Hughes, Douglas J Kojetin, John A Katzenellenbogen, Kendall W Nettles

Rapid on-chip genetic detection microfluidic platform for real world applications

用于实际应用的快速片上基因检测微流控平台

Senapati, Satyajyoti; Mahon, Andrew R; Gordon, Jason; Nowak, Carsten; Sengupta, Shramik; Powell, Thomas H Q; Feder, Jeffrey; Lodge, David M; Chang, Hsueh-Chia

CBP Is a dosage-dependent regulator of nuclear factor-kappaB suppression by the estrogen receptor

CBP 是一种剂量依赖性调节剂,可抑制雌激素受体对核因子 κB 的抑制

Kendall W Nettles, German Gil, Jason Nowak, Raphaël Métivier, Vandana B Sharma, Geoffrey L Greene