日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of Y-Shaped Covalent TEAD Inhibitors

基于结构的 Y 型共价 TEAD 抑制剂设计

Wenchao Lu, Mengyang Fan, Wenzhi Ji, Jason Tse, Inchul You, Scott B Ficarro, Isidoro Tavares, Jianwei Che, Audrey Y Kim, Xijun Zhu, Andrew Boghossian, Matthew G Rees, Melissa M Ronan, Jennifer A Roth, Stephen M Hinshaw, Behnam Nabet, Steven M Corsello, Nicholas Kwiatkowski, Jarrod A Marto, Tinghu Zh

Development of a Covalent Inhibitor of c-Jun N-Terminal Protein Kinase (JNK) 2/3 with Selectivity over JNK1

开发一种对 c-Jun N 端蛋白激酶 (JNK) 2/3 具有选择性而非 JNK1 的共价抑制剂

Wenchao Lu ,Yao Liu ,Yang Gao ,Qixiang Geng ,Deepak Gurbani ,Lianbo Li ,Scott B Ficarro ,Cynthia J Meyer ,Dhiraj Sinha ,Inchul You ,Jason Tse ,Zhixiang He ,Wenzhi Ji ,Jianwei Che ,Audrey Y Kim ,Tengteng Yu ,Kenneth Wen ,Kenneth C Anderson ,Jarrod A Marto ,Kenneth D Westover ,Tinghu Zhang ,Nathanael S Gray

Targeted kinase degradation via the KLHDC2 ubiquitin E3 ligase

通过 KLHDC2 泛素 E3 连接酶进行靶向激酶降解

Younghoon Kim, Pooreum Seo, Eunhye Jeon, Inchul You, Kyubin Hwang, Namkyoung Kim, Jason Tse, Juhyeon Bae, Ha-Soon Choi, Stephen M Hinshaw, Nathanael S Gray, Taebo Sim

Covalent disruptor of YAP-TEAD association suppresses defective Hippo signaling

YAP-TEAD 关联的共价破坏剂可抑制 Hippo 信号传导缺陷

Mengyang Fan #, Wenchao Lu #, Jianwei Che, Nicholas P Kwiatkowski, Yang Gao, Hyuk-Soo Seo, Scott B Ficarro, Prafulla C Gokhale, Yao Liu, Ezekiel A Geffken, Jimit Lakhani, Kijun Song, Miljan Kuljanin, Wenzhi Ji, Jie Jiang, Zhixiang He, Jason Tse, Andrew S Boghossian, Matthew G Rees, Melissa M Ronan, 

A Healthier Lifestyle Pattern for Cardiovascular Risk Reduction Is Associated With Better Bone Mass in Southern Chinese Elderly Men and Women

更健康的生活方式模式有助于降低心血管风险,并与中国南方老年男性和女性更好的骨密度相关。

Liu, Zhao-Min; Wong, Carmen Ka Man; Wong, Samuel Yeung-Shan; Leung, Jason; Tse, Lap Ah; Chan, Ruth; Woo, Jean