日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Parallel stopped-flow interrogation of diverse biological systems at the single-molecule scale

在单分子尺度上对多种生物系统进行并行停流分析

Kiselev, Roman; Brady, Ryan A; Modak, Arnab; Cruz-Navarrete, F Aaron; Alejo, Jose L; Terry, Daniel S; Altman, Roger B; Asher, Wesley B; Javitch, Jonathan A; Blanchard, Scott C

N-terminal fragment shedding contributes to signaling of the full-length adhesion receptor ADGRL3

N端片段脱落有助于全长粘附受体ADGRL3的信号传导。

Perry-Hauser, Nicole A; Du Rand, Jonathan R; Lee, Kuo Hao; Shi, Lei; Javitch, Jonathan A

Identification of a Lipid-Exposed Extrahelical Binding Site for Positive Allosteric Modulators of the Dopamine D(2) Receptor.

鉴定多巴胺 D(2) 受体正变构调节剂的脂质暴露螺旋外结合位点

Lim Herman D, Bartuzi Damian, Keen Alastair C, Rauffenbart Caroline, Glenn Jacqueline, Charlton Steven J, Lovera Silvia, Sands Zara A, Ates Ali, Wood Martyn, Canals Meritxell, Javitch Jonathan A, Carlsson Jens, Lane J Robert

Complex G-protein signaling of the adhesion GPCR, ADGRA3.

粘附 GPCR ADGRA3 的复杂 G 蛋白信号传导

Bagger Sofie M, Schihada Hannes, Walser Anna L S, Drzazga Anna K, Grätz Lukas, Palmisano Tiago, Kuhn Christina K, Mavri Maša, Mølleskov-Jensen Ann-Sophie, Tall Gregory G, Schöneberg Torsten, Mathiasen Signe J, Javitch Jonathan A, Schulte Gunnar, Spiess Katja, Rosenkilde Mette M

Habenular μ-opioid receptor knockout and chronic systemic receptor blockade promote negative affect and heighten nociceptive sensitivity

缰核μ-阿片受体敲除和慢性全身性受体阻滞会促进负面情绪并增强伤害感受敏感性。

Pekarskaya, Elizabeth A; Galiza Soares, Julia Alexsandra; Hough, Frances G; Langreck, Cory B; Tucciarone, Jason M; Javitch, Jonathan A

Conformational dynamics of the active state of β-arrestin 1

β-arrestin 1活性状态的构象动力学

Ngo, Van; Asher, Wesley B; Javitch, Jonathan A; Shi, Lei

CD33 and clusterin interact biophysically and genetically to modulate Alzheimer risk

CD33 和簇蛋白在生物物理和遗传学上相互作用,从而调节阿尔茨海默病风险。

Dodd, Roger B; Enomoto, Masahiro; Zhou, Ye; Satoh, Kanayo; Zhang, Yalun; Chen, Fusheng; Acheson, Beatrice; Ghaffari, Deniz; Sayn-Wittgenstein, Elizabeth; Manning, Jamie J; Dukas, George V; Patel, Ronak; Burguete, Alondra Schweizer; Kralovec, Mason J; Rashid, Mamunur; Hall, Jennifer L; Tamucci, Kirstin A; Chatila, Zena K; Liu, Minghua; Lee, Annie J; Vardarajan, Badri N; Taga, Mariko F; Pollari, Sirkku; Rabinovitch, Alon; Rillahan, Cory D; Bobkov, Andrey A; Sergienko, Eduard; Meadows, William; Qamar, Seema; Randle, Suzanne J; Johnson, Christopher M; Sevalle, Jean; Griffin, Jennifer; Bohm, Christopher; Ikura, Mitsuhiko; Xian, Xunde; Herz, Joachim; Kelly, Megan A; West, Jennifer; Satapathy, Sandeep; Wilson, Mark R; Javitch, Jonathan A; Fraser, Paul E; Bennett, David A; De Jager, Philip L; Fishelson, Zvi; Frenkel, Dan; Asher, Wesley B; Bradshaw, Elizabeth M; St George-Hyslop, Peter

Novel, small molecules targeting the 5-HT(4) receptor protect against stress-induced maladaptive behavior with efficacy across age

新型小分子靶向5-HT(4)受体,可有效预防各年龄段人群因应激引起的适应不良行为。

Ravenelle, Rebecca; Deng, Shi-Xian; Nelson, Mel; Pedersen, Maria H; Mendez-David, Indira; David, Denis J; Luna, Victor M; Turi, Gergely; Abramson, Madeline; Javitch, Jonathan A; Landry, Donald W; Chen, Briana K; Denny, Christine A

Altered striatal dopamine regulation in ADGRL3 knockout mice.

ADGRL3基因敲除小鼠纹状体多巴胺调节改变

Perry-Hauser Nicole A, Torres-Herraez Arturo, Boumhaouad Siham, Makowicz Emily A, Lowes Daniel C, Jin Michelle, Denny Christine A, Sulzer David, Mosharov Eugene V, Kellendonk Christoph, Javitch Jonathan A

Promiscuous G-protein activation by the calcium-sensing receptor

钙敏感受体对G蛋白的非特异性激活

Zuo, Hao; Park, Jinseo; Frangaj, Aurel; Ye, Jianxiang; Lu, Guanqi; Manning, Jamie J; Asher, Wesley B; Lu, Zhengyuan; Hu, Guo-Bin; Wang, Liguo; Mendez, Joshua; Eng, Edward; Zhang, Zhening; Lin, Xin; Grassucci, Robert; Hendrickson, Wayne A; Clarke, Oliver B; Javitch, Jonathan A; Conigrave, Arthur D; Fan, Qing R