Combined Scaffold Evaluation and Systems-Level Transcriptome-Based Analysis for Accelerated Lead Optimization Reveals Ribosomal Targeting Spirooxindole Cyclopropanes
结合支架评估和系统级转录组分析加速先导化合物优化,揭示核糖体靶向螺吲哚环丙烷
期刊:ChemMedChem
影响因子:3.6
doi:10.1002/cmdc.201900266
Kevin X Rodriguez, Erin N Howe, Emily P Bacher, Miranda Burnette, Jennifer L Meloche, Jayda Meisel, Patricia Schnepp, Xuejuan Tan, Mayland Chang, Jeremiah Zartman, Siyuan Zhang, Brandon L Ashfeld