CC-90009, a novel cereblon E3 ligase modulator, targets acute myeloid leukemia blasts and leukemia stem cells
CC-90009 是一种新型的 cereblon E3 连接酶调节剂,靶向急性髓系白血病原始细胞和白血病干细胞。
期刊:Blood
影响因子:23.1
doi:10.1182/blood.2020008676
Surka, Christine; Jin, Liqing; Mbong, Nathan; Lu, Chin-Chun; Jang, In Sock; Rychak, Emily; Mendy, Derek; Clayton, Thomas; Tindall, Elizabeth; Hsu, Christy; Fontanillo, Celia; Tran, Eileen; Contreras, Adrian; Ng, Stanley W K; Matyskiela, Mary; Wang, Kai; Chamberlain, Philip; Cathers, Brian; Carmichael, James; Hansen, Joshua; Wang, Jean C Y; Minden, Mark D; Fan, Jinhong; Pierce, Daniel W; Pourdehnad, Michael; Rolfe, Mark; Lopez-Girona, Antonia; Dick, John E; Lu, Gang