日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of an adenosquamous carcinoma histopathology - selective lung metastasis model

腺鳞癌组织病理学 - 选择性肺转移模型的开发

Iris A K Lähdeniemi, Jennifer R Devlin, Ashwini S Nagaraj, Sarang S Talwelkar, Jie Bao, Nora Linnavirta, Ceren Şeref Vujaklija, Elina A Kiss, Annabrita Hemmes, Emmy W Verschuren

The PP2A-Integrator-CDK9 axis fine-tunes transcription and can be targeted therapeutically in cancer

PP2A-Integrator-CDK9轴精细调控转录,可作为癌症治疗的靶点。

Stephin J Vervoort,Sarah A Welsh,Jennifer R Devlin,Elisa Barbieri,Deborah A Knight,Sarah Offley,Stefan Bjelosevic,Matteo Costacurta,Izabela Todorovski,Conor J Kearney,Jarrod J Sandow,Zheng Fan,Benjamin Blyth,Victoria McLeod,Joseph H A Vissers,Karolina Pavic,Ben P Martin,Gareth Gregory,Elena Demosthenous,Magnus Zethoven,Isabella Y Kong,Edwin D Hawkins,Simon J Hogg,Madison J Kelly,Andrea Newbold,Kaylene J Simpson,Otto Kauko,Kieran F Harvey,Michael Ohlmeyer,Jukka Westermarck,Nathanael Gray,Alessandro Gardini,Ricky W Johnstone

Targeting histone acetylation dynamics and oncogenic transcription by catalytic P300/CBP inhibition

通过抑制催化性P300/CBP来靶向组蛋白乙酰化动态和致癌转录

Simon J Hogg ,Olga Motorna ,Leonie A Cluse ,Timothy M Johanson ,Hannah D Coughlan ,Ramya Raviram ,Robert M Myers ,Matteo Costacurta ,Izabela Todorovski ,Lizzy Pijpers ,Stefan Bjelosevic ,Tobias Williams ,Shannon N Huskins ,Conor J Kearney ,Jennifer R Devlin ,Zheng Fan ,Jafar S Jabbari ,Ben P Martin ,Mohamed Fareh ,Madison J Kelly ,Daphné Dupéré-Richer ,Jarrod J Sandow ,Breon Feran ,Deborah Knight ,Tiffany Khong ,Andrew Spencer ,Simon J Harrison ,Gareth Gregory ,Vihandha O Wickramasinghe ,Andrew I Webb ,Phillippa C Taberlay ,Kenneth D Bromberg ,Albert Lai ,Anthony T Papenfuss ,Gordon K Smyth ,Rhys S Allan ,Jonathan D Licht ,Dan A Landau ,Omar Abdel-Wahab ,Jake Shortt ,Stephin J Vervoort ,Ricky W Johnstone

A novel CDK9 inhibitor increases the efficacy of venetoclax (ABT-199) in multiple models of hematologic malignancies

新型 CDK9 抑制剂可增强维奈克拉 (ABT-199) 在多种血液系统恶性肿瘤模型中的疗效

Darren C Phillips, Sha Jin, Gareth P Gregory, Qi Zhang, John Xue, Xiaoxian Zhao, Jun Chen, Yunsong Tong, Haichao Zhang, Morey Smith, Stephen K Tahir, Rick F Clark, Thomas D Penning, Jennifer R Devlin, Jake Shortt, Eric D Hsi, Daniel H Albert, Marina Konopleva, Ricky W Johnstone, Joel D Leverson, And

CDK13 cooperates with CDK12 to control global RNA polymerase II processivity

CDK13 与 CDK12 协同控制整体 RNA 聚合酶 II 的持续性

Zheng Fan, Jennifer R Devlin, Simon J Hogg, Maria A Doyle, Paul F Harrison, Izabela Todorovski, Leonie A Cluse, Deborah A Knight, Jarrod J Sandow, Gareth Gregory, Andrew Fox, Traude H Beilharz, Nicholas Kwiatkowski, Nichollas E Scott, Ana Tufegdzic Vidakovic, Gavin P Kelly, Jesper Q Svejstrup, Matth

Reprogrammed mRNA translation drives resistance to therapeutic targeting of ribosome biogenesis

重新编程的mRNA翻译驱动对核糖体生物合成治疗靶向性的抵抗

Eric P Kusnadi, Anna S Trigos, Carleen Cullinane, David L Goode, Ola Larsson, Jennifer R Devlin, Keefe T Chan, David P De Souza, Malcolm J McConville, Grant A McArthur, George Thomas, Elaine Sanij, Gretchen Poortinga, Ross D Hannan, Katherine M Hannan #, Jian Kang #, Richard B Pearson #

Inhibition of Pol I transcription treats murine and human AML by targeting the leukemia-initiating cell population

抑制 Pol I 转录可通过靶向白血病起始细胞群来治疗小鼠和人类 AML

Nadine Hein, Donald P Cameron, Katherine M Hannan, Nhu-Y N Nguyen, Chun Yew Fong, Jirawas Sornkom, Meaghan Wall, Megan Pavy, Carleen Cullinane, Jeannine Diesch, Jennifer R Devlin, Amee J George, Elaine Sanij, Jaclyn Quin, Gretchen Poortinga, Inge Verbrugge, Adele Baker, Denis Drygin, Simon J Harriso

Inhibition of RNA polymerase I transcription initiation by CX-5461 activates non-canonical ATM/ATR signaling

CX-5461 抑制 RNA 聚合酶 I 转录起始可激活非典型 ATM/ATR 信号

Jaclyn Quin, Keefe T Chan, Jennifer R Devlin, Donald P Cameron, Jeannine Diesch, Carleen Cullinane, Jessica Ahern, Amit Khot, Nadine Hein, Amee J George, Katherine M Hannan, Gretchen Poortinga, Karen E Sheppard, Kum Kum Khanna, Ricky W Johnstone, Denis Drygin, Grant A McArthur, Richard B Pearson, El

Combined inhibition of PI3K-related DNA damage response kinases and mTORC1 induces apoptosis in MYC-driven B-cell lymphomas

PI3K 相关 DNA 损伤反应激酶和 mTORC1 的联合抑制可诱导 MYC 驱动的 B 细胞淋巴瘤细胞凋亡

Jake Shortt, Benjamin P Martin, Andrea Newbold, Katherine M Hannan, Jennifer R Devlin, Adele J Baker, Rachael Ralli, Carleen Cullinane, Clemens A Schmitt, Maurice Reimann, Michael N Hall, Meaghan Wall, Ross D Hannan, Richard B Pearson, Grant A McArthur, Ricky W Johnstone