日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of HMGA2 inhibitors by AlphaScreen-based ultra-high-throughput screening assays

通过基于 AlphaScreen 的超高通量筛选试验鉴定 HMGA2 抑制剂

Linjia Su, Nadezda Bryan, Sabrina Battista, Juliano Freitas, Alyssa Garabedian, Federica D'Alessio, Miriam Romano, Fabiana Falanga, Alfredo Fusco, Lidia Kos, Jeremy Chambers, Francisco Fernandez-Lima, Prem P Chapagain, Stefan Vasile, Layton Smith, Fenfei Leng

Synthesis, biological evaluation, X-ray structure, and pharmacokinetics of aminopyrimidine c-jun-N-terminal kinase (JNK) inhibitors

氨基嘧啶 c-jun-N 端激酶 (JNK) 抑制剂的合成、生物学评价、X 射线结构和药代动力学

Ted Kamenecka, Rong Jiang, Xinyi Song, Derek Duckett, Weimin Chen, Yuan Yuan Ling, Jeff Habel, John D Laughlin, Jeremy Chambers, Mariana Figuera-Losada, Michael D Cameron, Li Lin, Claudia H Ruiz, Philip V LoGrasso