日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Glutathione responsive iNOS inhibiting polymeric prodrug for targeted Inhibition of angiogenesis

谷胱甘肽响应型iNOS抑制聚合物前药用于靶向抑制血管生成

Alimoradi, Houman; Fallah, Anita; Jespers, Pascale; Bolaky, Nargis; Gregoire, Françoise; Townley, Helen; Törnroth-Horsefield, Susanna; Shavandi, Armin; Dewachter, Laurence; Delporte, Christine

Doing More with Less: Accurate and Scalable Ligand Free Energy Calculations by Focusing on the Binding Site

以更少的资源实现更多目标:通过聚焦结合位点实现精确且可扩展的配体自由能计算

Alencar Araripe, David; Díaz-Holguín, Alejandro; Poso, Antti; van Westen, Gerard J P; Åqvist, Johan; Gutiérrez-de-Terán, Hugo; Jespers, Willem

Development of DuoMYC: a synthetic cell penetrant miniprotein that efficiently inhibits the oncogenic transcription factor MYC

DuoMYC的研发:一种能有效抑制致癌转录因子MYC的合成细胞穿透性小蛋白

Ellenbroek, Brecht D; Kahler, Jan Pascal; Arella, Damiano; Lin, Cherina; Jespers, Willem; Züger, Eliane Ann-Katrin; Drukker, Micha; Pomplun, Sebastian J

Large scale investigation of GPCR molecular dynamics data uncovers allosteric sites and lateral gateways

对GPCR分子动力学数据的大规模研究揭示了变构位点和侧向通道

Aranda-García, David; Stepniewski, Tomasz Maciej; Torrens-Fontanals, Mariona; García-Recio, Adrian; Lopez-Balastegui, Marta; Medel-Lacruz, Brian; Morales-Pastor, Adrián; Peralta-García, Alejandro; Dieguez-Eceolaza, Miguel; Sotillo-Nuñez, David; Ding, Tianyi; Drabek, Matthäus; Jacquemard, Célien; Jakowiecki, Jakub; Jespers, Willem; Jiménez-Rosés, Mireia; Jun-Yu-Lim, Víctor; Nicoli, Alessandro; Orzel, Urszula; Shahraki, Aida; Tiemann, Johanna K S; Ledesma-Martin, Vicente; Nerín-Fonz, Francho; Suárez-Dou, Sergio; Canal, Oriol; Pándy-Szekeres, Gáspár; Mao, Jiafei; Gloriam, David E; Kellenberger, Esther; Latek, Dorota; Guixà-González, Ramon; Gutiérrez-de-Terán, Hugo; Tikhonova, Irina G; Hildebrand, Peter W; Filizola, Marta; Babu, M Madan; Di Pizio, Antonella; Filipek, Slawomir; Kolb, Peter; Cordomi, Arnau; Giorgino, Toni; Marti-Solano, Maria; Selent, Jana

Accurate predictions of protein mutational effects accelerated with a hybrid-topology free energy protocol

利用混合拓扑自由能协议加速对蛋白质突变效应的精确预测

Koenekoop, Lucien; van de Brug, Nadine; Jespers, Willem; Åqvist, Johan; Gutiérrez-de-Terán, Hugo

Toward Assay-Aware Bioactivity Model(er)s: Getting a Grip on Biological Context

迈向基于检测的生物活性模型:把握生物学背景

Schoenmaker, Linde; Sastrokarijo, Enzo G; Heitman, Laura H; Beltman, Joost B; Jespers, Willem; van Westen, Gerard J P

In Search of Beautiful Molecules: A Perspective on Generative Modeling for Drug Design

探寻美丽的分子:药物设计生成建模的视角

van den Broek, Remco L; Patel, Shivam; van Westen, Gerard J P; Jespers, Willem; Sherman, Woody

HLA-E/peptide complexes differentially interact with NKG2A/CD94 and T cell receptors

HLA-E/肽复合物与NKG2A/CD94和T细胞受体的相互作用存在差异。

Voogd, Linda; van den Broek, Remco L; van Wolfswinkel, Marjolein; Franken, Kees L M C; Ruibal, Paula; Jespers, Willem; Leitner, Judith; Steinberger, Peter; van Westen, Gerard J P; Ottenhoff, Tom H M; Joosten, Simone A

Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools

探索新型地拉泽普衍生物作为hENT1抑制剂和潜在的共价分子工具

Dilweg, Majlen A; Gorostiola González, Marina; de Ruiter, Martijn D; Meijboom, Nadine J; van Veldhoven, Jacobus P D; Liu, Rongfang; Jespers, Willem; van Westen, Gerard J P; Heitman, Laura H; IJzerman, Adriaan P; van der Es, Daan

DIABEZE: Diabetes self-management among the elderly in a Belgian home for the aged: a best practice implementation project

DIABEZE:比利时养老院老年人糖尿病自我管理:最佳实践实施项目

Corremans, Marleen; Ohenewaa, Comfort; Van Steenberghe, Isaura; Bekkering, Trudy; Jespers, Hilke