Design, Synthesis and Biological Evaluation of Oxadiazole-Biphenyl Derivatives as Small Molecule Inhibitors Targeting PD-1/PD-L1 Immune Checkpoint
设计、合成及生物学评价恶二唑-联苯衍生物作为靶向PD-1/PD-L1免疫检查点的小分子抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.6c00048
Xie, Lingfeng; Zhu, Mingxuan; Zhao, Tong; Pei, Yifeng; Wei, Bo; Zhu, Shilong; Chen, Jiaoru; Zhang, Huibin; Zhou, Jinpei
PD-L1
Checkpoint
PD-1
免疫/内分泌