Discovery of Novel Quinoline-Based Proteasome Inhibitors for Human African Trypanosomiasis (HAT)
发现用于治疗人类非洲锥虫病(HAT)的新型喹啉类蛋白酶体抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c00791
Koester, Dennis C; Marx, Vanessa M; Williams, Sarah; Jiricek, Jan; Dauphinais, Maxime; René, Olivier; Miller, Sarah L; Zhang, Lei; Patra, Debjani; Chen, Yen-Liang; Cheung, Harry; Gable, Jonathan; Lakshminarayana, Suresh B; Osborne, Colin; Galarneau, Jean-Rene; Kulkarni, Upendra; Richmond, Wendy; Bretz, Angela; Xiao, Linda; Supek, Frantisek; Wiesmann, Christian; Honnappa, Srinivas; Be, Celine; Mäser, Pascal; Kaiser, Marcel; Ritchie, Ryan; Barrett, Michael P; Diagana, Thierry T; Sarko, Christopher; Rao, Srinivasa P S