日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

On-demand male contraception via acute inhibition of soluble adenylyl cyclase

通过急性抑制可溶性腺苷酸环化酶实现男性按需避孕

Melanie Balbach, Thomas Rossetti, Jacob Ferreira, Lubna Ghanem, Carla Ritagliati, Robert W Myers, David J Huggins, Clemens Steegborn, Ileana C Miranda, Peter T Meinke, Jochen Buck, Lonny R Levin

Architecture of androgen receptor pathways amplifying glucagon-like peptide-1 insulinotropic action in male pancreatic β cells

雄激素受体通路结构增强男性胰岛β细胞中胰高血糖素样肽-1的促胰岛素分泌作用

Weiwei Xu ,M M Fahd Qadir ,Daniela Nasteska ,Paula Mota de Sa ,Caroline M Gorvin ,Manuel Blandino-Rosano ,Charles R Evans ,Thuong Ho ,Evgeniy Potapenko ,Rajakrishnan Veluthakal ,Fiona B Ashford ,Stavroula Bitsi ,Jia Fan ,Manika Bhondeley ,Kejing Song ,Venkata N Sure ,Siva S V P Sakamuri ,Lina Schiffer ,Wandy Beatty ,Rachael Wyatt ,Daniel E Frigo ,Xiaowen Liu ,Prasad V Katakam ,Wiebke Arlt ,Jochen Buck ,Lonny R Levin ,Tony Hu ,Jay Kolls ,Charles F Burant ,Alejandra Tomas ,Matthew J Merrins ,Debbie C Thurmond ,Ernesto Bernal-Mizrachi ,David J Hodson ,Franck Mauvais-Jarvis

Design, Synthesis, and Pharmacological Evaluation of Second-Generation Soluble Adenylyl Cyclase (sAC, ADCY10) Inhibitors with Slow Dissociation Rates

具有慢解离速率的第二代可溶性腺苷酸环化酶 (sAC、ADCY10) 抑制剂的设计、合成及药理学评价

Michael Miller, Thomas Rossetti, Jacob Ferreira, Lubna Ghanem, Melanie Balbach, Navpreet Kaur, Lonny R Levin, Jochen Buck, Maria Kehr, Sandrine Coquille, Joop van den Heuvel, Clemens Steegborn, Makoto Fushimi, Efrat Finkin-Groner, Robert W Myers, Stacia Kargman, Nigel J Liverton, David J Huggins, Pe

Assessing potency and binding kinetics of soluble adenylyl cyclase (sAC) inhibitors to maximize therapeutic potential

评估可溶性腺苷酸环化酶 (sAC) 抑制剂的效力和结合动力学,以最大程度地发挥治疗潜力

Thomas Rossetti, Jacob Ferreira, Lubna Ghanem, Hannes Buck, Clemens Steegborn, Robert W Myers, Peter T Meinke, Lonny R Levin, Jochen Buck

Province-Wide Stool Color Card Screening for Biliary Atresia in Lower-Saxony: Experiences with Passive Distribution Strategies and Results

下萨克森州全省范围内开展胆道闭锁粪便颜色卡筛查:被动分发策略的经验和结果

Madadi-Sanjani, Omid; Kuebler, Joachim F; Uecker, Marie; Pfister, Eva-Doreen; Baumann, Ulrich; Kunze-Hullmann, Berit; Blaser, Jochen; Buck, Thomas; Petersen, Claus

Soluble adenylyl cyclase inhibition prevents human sperm functions essential for fertilization

可溶性腺苷酸环化酶抑制可阻止人类精子受精所必需的功能

Melanie Balbach, Lubna Ghanem, Thomas Rossetti, Navpreet Kaur, Carla Ritagliati, Jacob Ferreira, Dario Krapf, Lis C Puga Molina, Celia Maria Santi, Jan Niklas Hansen, Dagmar Wachten, Makoto Fushimi, Peter T Meinke, Jochen Buck, Lonny R Levin

Cholesterol Stabilizes TAZ in Hepatocytes to Promote Experimental Non-alcoholic Steatohepatitis

胆固醇稳定肝细胞中的TAZ以促进实验性非酒精性脂肪性肝炎

Xiaobo Wang, Bishuang Cai, Xiaoming Yang, Oluwatoni O Sonubi, Ze Zheng, Rajasekhar Ramakrishnan, Hongxue Shi, Luca Valenti, Utpal B Pajvani, Jaspreet Sandhu, Rodney E Infante, Arun Radhakrishnan, Douglas F Covey, Kun-Liang Guan, Jochen Buck, Lonny R Levin, Peter Tontonoz, Robert F Schwabe, Ira Tabas

Metabolic changes in mouse sperm during capacitation†

小鼠精子在获能过程中的代谢变化

Melanie Balbach, Maria Gracia Gervasi, David Martin Hidalgo, Pablo E Visconti, Lonny R Levin, Jochen Buck

Capacitation increases glucose consumption in murine sperm

获能增加小鼠精子的葡萄糖消耗

David M Hidalgo, Ana Romarowski, María G Gervasi, Felipe Navarrete, Melanie Balbach, Ana M Salicioni, Lonny R Levin, Jochen Buck, Pablo E Visconti

Mammalian pigmentation is regulated by a distinct cAMP-dependent mechanism that controls melanosome pH

哺乳动物的色素沉着受一种独特的cAMP依赖机制的调节,这种机制控制着黑素体的pH值

Dalee Zhou, Koji Ota, Charlee Nardin, Michelle Feldman, Adam Widman, Olivia Wind, Amanda Simon, Michael Reilly, Lonny R Levin, Jochen Buck, Kazumasa Wakamatsu, Shosuke Ito, Jonathan H Zippin