Synthesis and Pharmacological Characterization of Visabron, a Backbone Cyclic Peptide Dual Antagonist of α4β1 (VLA-4)/α9β1 Integrin for Therapy of Multiple Sclerosis
Visabron 的合成和药理学表征,一种用于治疗多发性硬化症的 α4β1 (VLA-4)/α9β1 整合素的骨架环肽双重拮抗剂
期刊:JACS Au
影响因子:8.5
doi:10.1021/jacsau.1c00496
Chaim Gilon, Michal Klazas, Adi Lahiani, Adi Schumacher-Klinger, Shira Merzbach, Johnny N Naoum, Haim Ovadia, Limor Rubin, Susan Cornell-Kennon, Erik M Schaefer, Jehoshua Katzhendler, Cezary Marcinkiewicz, Amnon Hoffman, Philip Lazarovici