日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological targeting of RIG-I can selectively activate the integrated stress response

通过药物靶向RIG-I可以选择性地激活整合应激反应。

Cuoco, Caroline A; Ren, Wen; Baron, Kelsey R; Gologo, Sakina; Perea, Valerie; Mathur, Prakhyat; Bora, Prerona; Ta, Amina; Chu, Alan; Aldakhlallah, Rama; Rhoades, Derek; Cole, Christian M; Tan, Ee Phie; Hou, William C; Yoon, Leonard; Guo, Xiaoyan; Rosarda, Jessica D; Baran, Phil S; Kampmann, Martin; Tillery, Lakeisha; Johnson, Kristen A; Powers, Evan T; Wiseman, R Luke; Kelly, Jeffery W

Autophagy activator AA-20 improves proteostasis and extends Caenorhabditis elegans lifespan

自噬激活剂AA-20改善蛋白质稳态并延长秀丽隐杆线虫的寿命

Tan, Ee Phie; Lyang, Nora; Doroodian, Saam; Sanz-Martinez, Pablo; Xu, Jin; Zaretski, Sviatlana; Nieto-Torres, José L; Ebata, Hiroshi; Lim, Shaun H Y; Hou, William C; Clay, Khalyd J; Yoon, Leonard; Massey, Lynée A; Rhoades, Derek; Garza, Danny; Johnson, Kristen A; To, Alan; Ambaye, Lydia; Bentley, Emily P; Petrascheck, Michael; Stolz, Alexandra; Kelly, Jeffery W; Hansen, Malene

Drug repurposing screen identifies an HRI activating compound that promotes adaptive mitochondrial remodeling in MFN2-deficient cells.

药物再利用筛选发现了一种 HRI 激活化合物,该化合物可促进 MFN2 缺陷细胞中的线粒体适应性重塑。

Bora Prerona, Zaman Mashiat, Oviedo Samantha, Kutseikin Sergei, Madrazo Nicole, Mathur Prakhyat, Pannikkat Meera, Krasny Sophia, Aldakhlallah Rama, Chu Alan, Johnson Kristen A, Grotjahn Danielle A, Shutt Timothy E, Wiseman R Luke

Targeted protein degradation by KLHDC2 ligands identified by high-throughput screening.

通过高通量筛选鉴定出KLHDC2配体对蛋白质的靶向降解作用

Zhou Han, Zhou Tonglian, Yu Wenli, Liu Liping, Ko Yeonjin, Johnson Kristen A, Wilson Ian A, Schultz Peter G, Bollong Michael J

Targeted Protein Degradation by KLHDC2 Ligands Identified by High Throughput Screening

高通量筛选鉴定出KLHDC2配体靶向降解蛋白质

Zhou, Han; Zhou, Tongliang; Yu, Wenli; Liu, Liping; Ko, Yeonjin; Johnson, Kristen A; Wilson, Ian A; Schultz, Peter G; Bollong, Michael J

Drug Repurposing Screen Identifies an HRI Activating Compound that Promotes Adaptive Mitochondrial Remodeling in MFN2-deficient Cells.

药物再利用筛选发现了一种 HRI 激活化合物,该化合物可促进 MFN2 缺陷细胞中的线粒体适应性重塑

Bora Prerona, Zaman Mashiat, Oviedo Samantha, Kutseikin Sergei, Madrazo Nicole, Mathur Prakhyat, Pannikkat Meera, Krasny Sophia, Chu Alan, Johnson Kristen A, Grotjahn Danielle A, Shutt Timothy E, Wiseman R Luke

Exploring Imaging Applications of a Red-Emitting π-Acceptor (π-A) Pyrene-Benzothiazolium Dye

探索红色发光π受体(π-A)芘-苯并噻唑鎓染料的成像应用

Abeywickrama, Chathura S; Huang, Enya; Yan, Wenhui; Vrionides, Michael A; Warushavithana, Paaramitha; Johnson, Kristen A; Stahelin, Robert V; Pang, Yi; Mani, Tomoyasu; Wijesinghe, Kaveesha J

Targeting FoxO transcription factors with HDAC inhibitors for the treatment of osteoarthritis

利用 HDAC 抑制剂靶向 FoxO 转录因子治疗骨关节炎

Ohzono, Hiroki; Hu, Yiwen; Nagira, Keita; Kanaya, Haruhisa; Okubo, Naoki; Olmer, Merissa; Gotoh, Masafumi; Kurakazu, Ichiro; Akasaki, Yukio; Kawata, Manabu; Chen, Emily; Chu, Alan C; Johnson, Kristen A; Lotz, Martin K

Pharmacological inhibition of CLK2 activates YAP by promoting alternative splicing of AMOTL2

CLK2 的药理学抑制通过促进 AMOTL2 的选择性剪接来激活 YAP。

Bulos, Maya L; Grzelak, Edyta M; Li-Ma, Chloris; Chen, Emily; Hull, Mitchell; Johnson, Kristen A; Bollong, Michael J

Measuring and Manipulating Membrane Cholesterol for the Study of Hedgehog Signaling

测量和操控膜胆固醇以研究 Hedgehog 信号通路

Kinnebrew, Maia; Johnson, Kristen A; Radhakrishnan, Arun; Rohatgi, Rajat