日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Compounds Reducing Human Sperm Motility as Potential Nonhormonal Contraceptives Identified Using a High-Throughput Phenotypic Screening Platform

利用高通量表型筛选平台鉴定出可降低人类精子活力的化合物,这些化合物有望成为非激素避孕药。

Richardson, Anthony; Gruber, Franz S; Day, David P; Edwards, Darren; Georgiou, Irene; Johnston, Zoe C; Joji, Halimatu; Martins da Silva, Sarah; Myles, Rachel; Norcross, Neil R; Read, Kevin D; Swedlow, Jason R; Wilson, Caroline; Barratt, Christopher L R; Gilbert, Ian H

Rational Exploration of 2,4-Diaminopyrimidines as DHFR Inhibitors Active against Mycobacterium abscessus and Mycobacterium avium, Two Emerging Human Pathogens.

合理探索 2,4-二氨基嘧啶作为 DHFR 抑制剂对脓肿分枝杆菌和鸟分枝杆菌(两种新兴人类病原体)的活性

Andrade Meirelles Matheus, Almeida Vitor M, Sullivan Jaryd R, de Toledo Ian, Dos Reis Caio Vinicius, Cunha Micael Rodrigues, Zigweid Rachel, Shim Abraham, Sankaran Banumathi, Woodward Elijah L, Seibold Steve, Liu Lijun, Mian Mohammad Rasel, Battaile Kevin P, Riley Jennifer, Duncan Christina, Simeons Frederick R C, Ferguson Liam, Joji Halimatu, Read Kevin D, Lovell Scott, Staker Bart L, Behr Marcel A, Pilli Ronaldo A, Couñago Rafael M

Identification of a potent and selective LAPTc inhibitor by RapidFire-Mass Spectrometry, with antichagasic activity

利用快速质谱法鉴定出一种高效且选择性的LAPTc抑制剂,该抑制剂具有抗锥虫病活性。

Izquierdo, Maikel; Lin, De; O'Neill, Sandra; Webster, Lauren A; Paterson, Christy; Thomas, John; Aguado, Mirtha Elisa; Colina Araújo, Enrique; Alpízar-Pedraza, Daniel; Joji, Halimatu; MacLean, Lorna; Hope, Anthony; Gray, David W; Zoltner, Martin; Field, Mark C; González-Bacerio, Jorge; De Rycker, Manu