Development of Dimethylisoxazole-Attached Imidazo[1,2- a]pyridines as Potent and Selective CBP/P300 Inhibitors
二甲基异恶唑连接的咪唑并[1,2- a]吡啶作为有效和选择性 CBP/P300 抑制剂的开发
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.0c02232
Alex Muthengi, Virangika K Wimalasena, Hailemichael O Yosief, Melissa J Bikowitz, Logan H Sigua, Tingjian Wang, Deyao Li, Zied Gaieb, Gagan Dhawan, Shuai Liu, Jon Erickson, Rommie E Amaro, Ernst Schönbrunn, Jun Qi, Wei Zhang