High-affinity small-molecule inhibitors of the menin-mixed lineage leukemia (MLL) interaction closely mimic a natural protein-protein interaction
高亲和力的小分子抑制剂能够有效抑制menin-混合谱系白血病(MLL)相互作用,并高度模拟天然蛋白质-蛋白质相互作用。
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm401868d
Shihan He ,Timothy J Senter, Jonathan Pollock, Changho Han, Sunil Kumar Upadhyay, Trupta Purohit, Rocco D Gogliotti, Craig W Lindsley, Tomasz Cierpicki, Shaun R Stauffer, Jolanta Grembecka