日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A degron-mimicking molecular glue drives CRBN homo-dimerization and degradation.

类似降解子的分子胶驱动 CRBN 同源二聚化和降解。

Langousis Gerasimos, Gainza Pablo, Hunkeler Moritz, Kapsitidou Despoina, Donckele Etienne J, Annunziato Stefano, Wiedmer Lars, Jones Katherine F M, DeMarco Bradley, Quan Chao, Bunker Richard D, Lumb Kevin J, Fasching Bernhard, Castle John C, Townson Sharon A, Bonenfant Débora

Targeting N-Myc in neuroblastoma with selective Aurora kinase A degraders.

利用选择性 Aurora 激酶 A 降解剂靶向神经母细胞瘤中的 N-Myc

Tang Jian, Moorthy Ramkumar, Hirsch Laura E, Demir Özlem, Baker Zachary D, Naumann Jordan A, Jones Katherine F M, Grillo Michael J, Haefner Ella S, Shi Ke, Levy Michaella J, Gupta Harshita B, Aihara Hideki, Harris Reuben S, Amaro Rommie E, Levinson Nicholas M, Harki Daniel A

Development of Allosteric Small Molecule APOBEC3B Inhibitors from In Silico Screening

基于计算机筛选的变构小分子APOBEC3B抑制剂的开发

Jones, Katherine F M; Demir, Özlem; Wyllie, Mackenzie K; Grillo, Michael J; Morris, Clare; Hirakis, Sophia P; Kardile, Rahul Dadabhau; Walters, Michael A; Harris, Reuben S; Amaro, Rommie E; Harki, Daniel A

APOBEC3A Catalytic Inactivity Mutation Induces Tertiary Structure Destabilization

APOBEC3A催化失活突变导致三级结构不稳定

Jones, Katherine F M; Shehata, Mohamed; Carpenter, Michael A; Amaro, Rommie E; Harki, Daniel A

The current toolbox for APOBEC drug discovery

APOBEC药物发现的现有工具箱

Grillo, Michael J; Jones, Katherine F M; Carpenter, Michael A; Harris, Reuben S; Harki, Daniel A