日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Expanding the druggable zinc-finger proteome defines properties of drug-induced degradation.

扩大可成药锌指蛋白组,可以明确药物诱导降解的特性

Słabicki Mikołaj, Park Jiho, Nowak Radosław P, Roy Burman Shourya S, Pellman Jesse, Zou Charles, Razumkov Hlib, Carreiro Jeannie, Rastogi Simran, Goldstein Anna, Nagiec Marek M, Donovan Katherine A, Che Jianwei, Hunkeler Moritz, Geng Qixiang, Hsu Chi-Lin, Lakshminarayan Megha, Shu Chelsea, Zon Rebecca L, Kozicka Zuzanna, Park Paul M C, Tsai Jonathan M, Yoon Hojong, Jones Lyn H, Sperling Adam S, Gray Nathanael S, Fischer Eric S, Ebert Benjamin L

Advances in sulfonyl exchange chemical biology: expanding druggable target space

磺酰交换化学生物学的进展:拓展药物靶点空间

Jones, Lyn H

Property-Based Optimization of Cereblon-Based Molecular Glue Degraders

基于性质的塞雷布隆基分子胶降解剂的优化

Jones, Lyn H

Structure-guided design of a truncated heterobivalent chemical probe degrader of IRE1α

基于结构的截短型异二价化学探针IRE1α降解剂的设计

Zerfas, Breanna L; Liu, Yingpeng; Che, Jianwei; Donovan, Katherine A; Hatcher, John M; Huerta, Fidel; Metivier, Rebecca J; Nowak, Radosław P; Ragosta, Leah; Tsang, Tiffany; Fischer, Eric S; Jones, Lyn H

Introduction to the themed collection on 'Induced-Proximity Pharmacology'

“诱导邻近药理学”主题系列介绍

Hartung, Ingo V; James, Lindsey I; Jones, Lyn H

The Minimum Protein Staple? - Towards 'bio'-Baldwin's rules via inter-phosphosite linking in the MEK1 activation loop

最低限度的蛋白质必需成分?——通过MEK1激活环中的磷酸化位点间连接,迈向“生物”鲍德温规则

Galan, Sébastien R G; Raj, Ritu; Mamalis, Dimitrios; Jones, Lyn H; Mohammed, Shabaz; Davis, Benjamin G

Development of sulfonyl fluoride chemical probes to advance the discovery of cereblon modulators

开发磺酰氟化学探针以推进脑蛋白调节剂的发现

Liu, Yingpeng; Nowak, Radosław P; Che, Jianwei; Donovan, Katherine A; Huerta, Fidel; Liu, Hu; Metivier, Rebecca J; Fischer, Eric S; Jones, Lyn H

Synthetic modification of protein surfaces to mediate induced-proximity pharmacology

通过对蛋白质表面进行合成修饰来介导诱导邻近药理学

Jones, Lyn H

Catalytic Degraders Effectively Address Kinase Site Mutations in EML4-ALK Oncogenic Fusions

催化降解剂可有效解决EML4-ALK致癌融合蛋白中的激酶位点突变

Gao, Yang; Jiang, Baishan; Kim, Hellen; Berberich, Matthew J; Che, Jianwei; Donovan, Katherine A; Hatcher, John M; Huerta, Fidel; Kwiatkowski, Nicholas P; Liu, Yingpeng; Liuni, Peter P; Metivier, Rebecca J; Murali, Vineeth K; Nowak, Radosław P; Zhang, Tinghu; Fischer, Eric S; Gray, Nathanael S; Jones, Lyn H

Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange

利用硫杂环交换法对 Cereblon 传感器环组氨酸进行共价交联

Cruite, Justin T; Nowak, Radosław P; Donovan, Katherine A; Ficarro, Scott B; Huang, Huang; Liu, Hu; Liu, Yingpeng; Marto, Jarrod A; Metivier, Rebecca J; Fischer, Eric S; Jones, Lyn H