日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of mCMV280: An Oral Ectoparasiticide in the Isoxazoline Class with Reduced Mammalian Brain Exposure

mCMV280 的发现:一种异噁唑啉类口服体外寄生虫杀灭剂,可降低哺乳动物大脑暴露量

McComic, Sarah E; Wilson, Katy B; Li, Zhilin; Chen, Jeffrey; Weiss, Frank; Song, Lirui; Mazumdar, Wrickban; Dvorak, Curt A; Brittain, Jason; Lee, Kyoung-Jin; Li, Shuangwei; Joseph, Sean B; McNamara, Case W; Vos, Martijn W; Sheshachalam, Avinash; Inácio, Alex; Dechering, Koen J; Chatterjee, Arnab K; Swale, Daniel R

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

A drug repurposing approach reveals targetable epigenetic pathways in Plasmodium vivax hypnozoites.

药物再利用方法揭示了间日疟原虫休眠子中可靶向的表观遗传通路

Maher Steven P, Bakowski Malina A, Vantaux Amélie, Flannery Erika L, Andolina Chiara, Gupta Mohit, Antonova-Koch Yevgeniya, Argomaniz Magdalena, Cabrera-Mora Monica, Campo Brice, Chao Alexander T, Chatterjee Arnab K, Cheng Wayne T, Chuenchob Vorada, Cooper Caitlin A, Cottier Karissa, Galinski Mary R, Harupa-Chung Anke, Ji Hana, Joseph Sean B, Lenz Todd, Lonardi Stefano, Matheson Jessica, Mikolajczak Sebastian A, Moeller Timothy, Orban Agnes, Padín-Irizarry Vivian, Pan Kastin, Péneau Julie, Prudhomme Jacques, Roesch Camille, Ruberto Anthony, Sabnis Saniya S, Saney Celia L, Sattabongkot Jetsumon, Sereshki Saleh, Suriyakan Sangrawee, Ubalee Ratawan, Wang Yinsheng, Wasisakun Praphan, Yin Jiekai, Popovici Jean, McNamara Case W, Joyner Chester, Nosten François H, Witkowski Benoît, Le Roch Karine G, Kyle Dennis E

The Transformative Impact of the African Cohort Study (AFRICOS) Toward Reaching HIV 95-95-95 Goals in Sub-Saharan Africa

非洲队列研究(AFRICOS)对撒哈拉以南非洲实现艾滋病毒95-95-95目标的变革性影响

Shah, Neha; Crowell, Trevor A; Hern, Jaclyn; Anyebe, Victor; Bahemana, Emmanuel; Kibuuka, Hannah; Singoei, Valentine; Maswai, Jonah; Parikh, Ajay; Duff, Emma R; Cavanaugh, Joseph Sean; Romo, Matthew L; Ake, Julie A; Reid, Michael J A; Nkengasong, Amb John N

NK2R signaling governs intestinal lipid mobilization and mucosal inflammation

NK2R信号通路调控肠道脂质动员和黏膜炎症。

Perez, Pedro A; Liu, Chung-Chih; Ferrari, Alessandra; Littlejohn, Nicole; Kennelly, John Paul; Robinson, Emma; Nguyen-Tran, Vân T B; Athanacio, Jon; Joseph, Sean B; Amso, Zaid; Tontonoz, Peter; Srinivasan, Supriya

Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead

CMX990 的发现:一种带有新型弹头的强效 SARS-CoV-2 3CL 蛋白酶抑制剂

Dayan Elshan, N G R; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

Correction to "Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead"

对“CMX990的发现:一种带有新型弹头的强效SARS-CoV-2 3CL蛋白酶抑制剂”一文的更正

Elshan, N G R Dayan; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Liu, Dongdong; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

A small molecule MST1/2 inhibitor accelerates murine liver regeneration with improved survival in models of steatohepatitis.

小分子 MST1/2 抑制剂可加速小鼠肝脏再生,提高脂肪性肝炎模型小鼠的存活率

Watkins Ryan, Gamo Ana, Choi Seung Hyuk, Kumar Manoj, Buckarma EeeLN, McCabe Chantal, Tomlinson Jennifer, Pereya David, Lupse Blaz, Geravandi Shirin, Werneburg Nathan W, Wang Chen, Starlinger Patrick, Zhu Siying, Li Sijia, Yu Shan, Surakattula Murali, Baguley Tyler, Ardestani Amin, Maedler Kathrin, Roland Jason, Nguyen-Tran Van, Joseph Sean, Petrassi Mike, Rogers Nikki, Gores Gregory, Chatterjee Arnab, Tremblay Matthew, Shen Weijun, Smoot Rory

Pharmacokinetics and Pharmacodynamics of Clofazimine for Treatment of Cryptosporidiosis

氯法齐明治疗隐孢子虫病的药代动力学和药效学研究

Zhang, Cindy X; Love, Melissa S; McNamara, Case W; Chi, Victor; Woods, Ashley K; Joseph, Sean; Schaefer, Deborah A; Betzer, Dana P; Riggs, Michael W; Iroh Tam, Pui-Ying; Van Voorhis, Wesley C; Arnold, Samuel L M

Ozone-induced enhancement of airway hyperreactivity in rhesus macaques: Effects of antioxidant treatment

臭氧诱导恒河猴气道高反应性的增强:抗氧化剂治疗的影响

Cameron H Flayer, Erik D Larson, Anjali Joseph, Sean Kao, Wenxiu Qu, Austin Van Haren, Christopher M Royer, Lisa A Miller, John P Capitanio, Thais Sielecki, Melpo Christofidou-Solomidou, Angela Haczku