Use of a Conformational-Switching Mechanism to Modulate Exposed Polarity: Discovery of CCR2 Antagonist BMS-741672
利用构象转换机制调节暴露极性:CCR2拮抗剂BMS-741672的发现
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.8b00439
Yang, Michael G; Xiao, Zili; Cherney, Robert J; Tebben, Andrew J; Batt, Douglas G; Brown, Gregory D; Chen, Jing; Cvijic, Mary Ellen; Dabros, Marta; Duncia, John V; Galella, Michael; Gardner, Daniel S; Khandelwal, Purnima; Ko, Soo S; Malley, Mary F; Mo, Ruowei; Pang, Jian; Rose, Anne V; Santella, Joseph B 3rd; Shi, Hong; Srivastava, Anurag; Traeger, Sarah C; Wang, Bei; Xu, Songmei; Zhao, Rulin; Barrish, Joel C; Mandlekar, Sandhya; Zhao, Qihong; Carter, Percy H