Structure-Guided Synthesis of FK506 and FK520 Analogs with Increased Selectivity Exhibit In Vivo Therapeutic Efficacy against Cryptococcus
结构引导合成选择性更高的 FK506 和 FK520 类似物,在体内表现出对隐球菌的治疗效果
期刊:mBio
影响因子:5.1
doi:10.1128/mbio.01049-22
Michael J Hoy, Eunchong Park #, Hyunji Lee #, Won Young Lim #, D Christopher Cole, Nicholas D DeBouver, Benjamin G Bobay, Phillip G Pierce, David Fox 3rd, Maria Ciofani, Praveen R Juvvadi, William Steinbach, Jiyong Hong, Joseph Heitman