Phage-assisted, active site-directed ligand evolution of a potent and selective histone deacetylase 8 inhibitor
利用噬菌体辅助的活性位点定向配体进化方法,开发出一种高效且选择性的组蛋白去乙酰化酶 8 抑制剂
期刊:Protein Science
影响因子:5.2
doi:10.1002/pro.4512
Morse, Jared S; Sheng, Yan J; Hampton, Joshua Trae; Sylvain, Lauralee D; Das, Sukant; Alugubelli, Yugendar R; Chen, Peng-Hsun Chase; Yang, Kai S; Xu, Shiqing; Fierke, Carol A; Liu, Wenshe Ray