日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule-constrained paratope mimetic bicyclic peptides as potent inhibitors of group 1 and 2 influenza A virus hemagglutinins

小分子约束的互补位模拟双环肽作为1组和2组甲型流感病毒血凝素的强效抑制剂

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Garg, Divita; Zhu, Xueyong; Jongeneelen, Mandy; Tang, Chan; Schepens, Wim B G; Buyck, Christophe; Stoops, Bart; Vermond, Jan; Vogels, Ronald; Friesen, Robert H E; van Dongen, Maria J P; Wilson, Ian A

AI-guided prefusion stabilization of the human coronavirus OC43 spike protein enables universal embecovirus antigen design

人工智能引导的人类冠状病毒OC43刺突蛋白融合前稳定化技术实现了通用型恩贝病毒抗原设计

Melchers, Jelle M; Juraszek, Jarek; Hulswit, Ruben J G; van Overveld, Daan; Le, Lam; van Kuppeveld, Frank J M; Hurdiss, Daniel L; Bosch, Berend-Jan; Langedijk, Johannes P M; Bakkers, Mark J G

De novo design of D-peptide ligands: Application to influenza virus hemagglutinin.

从头设计 D 肽配体:应用于流感病毒血凝素

Juraszek Jarek, Kadam Rameshwar U, Branduardi Davide, van Ameijde Jeroen, Garg Divita, Dailly Nicolas, Jongeneelen Mandy, Vermond Jan, Brakenhoff Just P J, Brandenburg Boerries, van Dongen Maria J P, Vogels Ronald, Friesen Robert H E, Wilson Ian A

V(H)H antibody loop guides design of a synthetic macrocyclic peptide that potently blocks influenza virus membrane fusion

V(H)H抗体环指导合成大环肽的设计,该大环肽能有效阻断流感病毒膜融合。

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Garg, Divita; Zhu, Xueyong; Jongeneelen, Mandy; Schepens, Wim B G; Stoops, Bart; Vermond, Jan; Goutier, Wouter; Tang, Chan; Blokland, Sven; Vogels, Ronald; Friesen, Robert H E; van Dongen, Maria J P; Wilson, Ian A

Absolute quantitation of binding antibodies from clinical samples

临床样本中结合抗体的绝对定量

Tang, Chan; Verwilligen, Annemiek; Sadoff, Jerald; Brandenburg, Boerries; Sneekes-Vriese, Eveline; van den Kerkhof, Tom; Dillen, Lieve; Rutten, Lucy; Juraszek, Jarek; Callewaert, Katleen; Janssen, Sarah; Huizingh, Jeroen; Euler, Zelda; Schilperoord, Tom; Verhemeldonck, Marc; Langedijk, Johannes P M; Hendriks, Jenny; Stieh, Daniel J

Impact of SARS-CoV-2 spike stability and RBD exposure on antigenicity and immunogenicity

SARS-CoV-2刺突蛋白稳定性及RBD暴露对抗原性和免疫原性的影响

Rutten, Lucy; Swart, Maarten; Koornneef, Annemart; Bouchier, Pascale; Blokland, Sven; Sadi, Ava; Juraszek, Jarek; Vijayan, Aneesh; Schmit-Tillemans, Sonja; Verspuij, Johan; Choi, Ying; Daal, Chenandly E; Perkasa, Aditya; Torres Morales, Shessy; Myeni, Sebenzile K; Kikkert, Marjolein; Tolboom, Jeroen; van Manen, Daniëlle; Kuipers, Harmjan; Schuitemaker, Hanneke; Zahn, Roland; Langedijk, Johannes P M

Potent peptidic fusion inhibitors of influenza virus

流感病毒的强效肽融合抑制剂

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Buyck, Christophe; Schepens, Wim B G; Kesteleyn, Bart; Stoops, Bart; Vreeken, Rob J; Vermond, Jan; Goutier, Wouter; Tang, Chan; Vogels, Ronald; Friesen, Robert H E; Goudsmit, Jaap; van Dongen, Maria J P; Wilson, Ian A

(Un)Folding mechanisms of the FBP28 WW domain in explicit solvent revealed by multiple rare event simulation methods

利用多种稀有事件模拟方法揭示FBP28 WW结构域在显式溶剂中的(解)折叠机制

Juraszek, Jarek; Bolhuis, Peter G