Biochemical Characterization and Structure-Based Mutational Analysis Provide Insight into the Binding and Mechanism of Action of Novel Aspartate Aminotransferase Inhibitors
生化表征和基于结构的突变分析为新型天冬氨酸氨基转移酶抑制剂的结合和作用机制提供了见解
期刊:Biochemistry
影响因子:2.9
doi:10.1021/acs.biochem.8b00914
Melissa C Holt, Zahra Assar, Reza Beheshti Zavareh, Lin Lin, Justin Anglin, Oksana Mashadova, Daniel Haldar, Edouard Mullarky, Daniel M Kremer, Lewis C Cantley, Alec C Kimmelman, Adam J Stein, Luke L Lairson, Costas A Lyssiotis