日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural basis of SARS-CoV-2 polymerase inhibition by nonnucleoside inhibitor HeE1-2Tyr

非核苷类抑制剂HeE1-2Tyr抑制SARS-CoV-2聚合酶的结构基础

Kabinger, Florian; Doze, Valerie; Schmitzová, Jana; Lidschreiber, Michael; Dienemann, Christian; Cramer, Patrick

Targeted degradation of CDK9 potently disrupts the MYC-regulated network.

靶向降解 CDK9 可有效破坏 MYC 调控网络

Toure Mohammed A, Motoyama Keisuke, Xiang Yichen, Urgiles Julie, Kabinger Florian, Koglin Ann-Sophie, Iyer Ramya S, Gagnon Kaitlyn, Kumar Amruth, Ojeda Samuel, Harrison Drew A, Rees Matthew G, Roth Jennifer A, Ott Christopher J, Schiavoni Richard, Whittaker Charles A, Levine Stuart S, White Forest M, Calo Eliezer, Richters Andre, Koehler Angela N

Tail-tape-fused virion and non-virion RNA polymerases of a thermophilic virus with an extremely long tail

具有极长尾巴的嗜热病毒的尾带融合病毒体和非病毒体 RNA 聚合酶

Anastasiia Chaban #, Leonid Minakhin #, Ekaterina Goldobina, Brain Bae, Yue Hao, Sergei Borukhov, Leena Putzeys, Maarten Boon, Florian Kabinger, Rob Lavigne, Kira S Makarova, Eugene V Koonin, Satish K Nair, Shunsuke Tagami, Konstantin Severinov, Maria L Sokolova

Mechanism of molnupiravir-induced SARS-CoV-2 mutagenesis

莫努匹拉韦诱发 SARS-CoV-2 突变的机制

Florian Kabinger #, Carina Stiller #, Jana Schmitzová #, Christian Dienemann, Goran Kokic, Hauke S Hillen, Claudia Höbartner, Patrick Cramer

Modulating Androgen Receptor-Driven Transcription in Prostate Cancer with Selective CDK9 Inhibitors

使用选择性 CDK9 抑制剂调节前列腺癌中的雄激素受体驱动的转录

André Richters, Shelby K Doyle, David B Freeman, Christina Lee, Becky S Leifer, Sajjeev Jagannathan, Florian Kabinger, Jošt Vrabič Koren, Nicholas B Struntz, Julie Urgiles, Ryan A Stagg, Brice H Curtin, Deep Chatterjee, Sebastian Mathea, Peter J Mikochik, Tamara D Hopkins, Hua Gao, Jonathan R Branch