日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CRM1 regulates androgen receptor stability and impacts DNA repair pathways in prostate cancer, independent of the androgen receptor.

CRM1 调节雄激素受体的稳定性,并影响前列腺癌中的 DNA 修复途径,而与雄激素受体无关

Kumar Rajendra, Mendonca Janet, Shetty Abhishek, Yang Yuhan, Owoyemi Olutosin, Wilson Lillian, Boyapati Kavya, Topiwala Deven, Thomas Naiju, Nguyen Huong, Luo Jun, Paller Channing J, Denmeade Samuel R, Carducci Michael A, Kachhap Sushant K

Phase I Trial of Intravenous Mistletoe Extract in Advanced Cancer

晚期癌症患者静脉注射槲寄生提取物的I期临床试验

Paller, Channing J; Wang, Lin; Fu, Wei; Kumar, Rajendra; Durham, Jennifer N; Azad, Nilofer S; Laheru, Daniel A; Browner, Ilene; Kachhap, Sushant K; Boyapati, Kavya; Odeny, Thomas; Armstrong, Deborah K; Meyer, Christian F; Gaillard, Stephanie; Brahmer, Julie R; Page, Ivelisse; Wang, Hao; Diaz, Luis A Jr

Supraphysiologic Testosterone Induces Ferroptosis and Activates Immune Pathways through Nucleophagy in Prostate Cancer

超生理水平的睾酮通过核自噬诱导前列腺癌细胞发生铁死亡并激活免疫通路

Kumar, Rajendra; Mendonca, Janet; Owoyemi, Olutosin; Boyapati, Kavya; Thomas, Naiju; Kanacharoen, Suthicha; Coffey, Max; Topiwala, Deven; Gomes, Carolina; Ozbek, Busra; Jones, Tracy; Rosen, Marc; Dong, Liang; Wiens, Sadie; Brennen, W Nathaniel; Isaacs, John T; De Marzo, Angelo M; Markowski, Mark C; Antonarakis, Emmanuel S; Qian, David Z; Pienta, Kenneth J; Pardoll, Drew M; Carducci, Michael A; Denmeade, Samuel R; Kachhap, Sushant K

HIF1 and ID1 Interplay Confers Adaptive Survival to HIF1α-Inhibition

HIF1和ID1的相互作用赋予HIF1α抑制适应性生存能力

Geng, Hao; Ko, Hyun-Kyung; Pittsenbarger, Janet; Harvey, Christopher T; Xue, Changhui; Liu, Qiong; Wiens, Sadie; Kachhap, Sushant K; Beer, Tomasz M; Qian, David Z

Small-molecule screening of PC3 prostate cancer cells identifies tilorone dihydrochloride to selectively inhibit cell growth based on cyclin-dependent kinase 5 expression

对PC3前列腺癌细胞进行小分子筛选,发现盐酸替洛酮能够基于细胞周期蛋白依赖性激酶5的表达选择性地抑制细胞生长。

Wissing, Michel D; Dadon, Tikva; Kim, Eunice; Piontek, Klaus B; Shim, Joong S; Kaelber, Nadine S; Liu, Jun O; Kachhap, Sushant K; Nelkin, Barry D

Repurposing itraconazole as a treatment for advanced prostate cancer: a noncomparative randomized phase II trial in men with metastatic castration-resistant prostate cancer

将伊曲康唑重新用于治疗晚期前列腺癌:一项针对转移性去势抵抗性前列腺癌患者的非对照随机II期试验

Antonarakis, Emmanuel S; Heath, Elisabeth I; Smith, David C; Rathkopf, Dana; Blackford, Amanda L; Danila, Daniel C; King, Serina; Frost, Anja; Ajiboye, A Seun; Zhao, Ming; Mendonca, Janet; Kachhap, Sushant K; Rudek, Michelle A; Carducci, Michael A

Downregulation of homologous recombination DNA repair genes by HDAC inhibition in prostate cancer is mediated through the E2F1 transcription factor

前列腺癌中 HDAC 抑制剂通过 E2F1 转录因子介导同源重组 DNA 修复基因的下调,从而导致同源重组 DNA 修复基因表达下调。

Kachhap, Sushant K; Rosmus, Nadine; Collis, Spencer J; Kortenhorst, Madeleine S Q; Wissing, Michel D; Hedayati, Mohammad; Shabbeer, Shabana; Mendonca, Janet; Deangelis, Justin; Marchionni, Luigi; Lin, Jianqing; Höti, Naseruddin; Nortier, Johan W R; DeWeese, Theodore L; Hammers, Hans; Carducci, Michael A