日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Scaffold Fusion and SAR Transfer with a Chemical Language Model Generates Novel Liver X Receptor Modulators

利用化学语言模型进行支架融合和构效关系转移,生成新型肝X受体调节剂

Bandomir, Nils Christiaan; Hörmann, Tim; Kärcher, Annette; Kaiser, Astrid; Merk, Daniel; Heitel, Pascal

Structure-Based Design of PROTACS for the Degradation of Soluble Epoxide Hydrolase.

基于结构的PROTACS设计用于降解可溶性环氧化物水解酶

Schönfeld Julia, Brunst Steffen, Ciomirtan Ludmila, Willmer Lena, Chromik Michel A, Kumar Adarsh, Froemel Timo, Liebisch Nick, Hackspacher Arne, Ehrler Johanna H M, Wintermeier Lukas, Hesse Christina, Fiedler Jan, Heering Jan, Freitag Hinrich, Zardo Patrick, Fieguth Hans-Gerd, Brüggerhoff Astrid, Jakob Josefine, Häupl Björn, Weizel Lilia, Kaiser Astrid, Schubert-Zsilavecz Manfred, Oellerich Thomas, Fleming Ingrid, Schebb Nils H, Fürst Robert, Kannt Aimo, Knapp Stefan, Proschak Ewgenij, Hiesinger Kerstin

Fragment-Based Discovery of Drug-like LRH-1 Agonists

基于片段的类药LRH-1激动剂发现

Lang, Alisa; Ildefeld, Niklas; Lillich, Felix F; Kaiser, Astrid; Busch, Romy; Marschner, Julian A; Proschak, Ewgenij; Heering, Jan; Schubert-Zsilavecz, Manfred; Merk, Daniel

Efficacy of MP1032 in hospitalised patients with COVID-19- authors' reply

MP1032治疗COVID-19住院患者的疗效——作者回复

Sager, Petra; Kaiser, Astrid; Schumann, Sara; Ludescher, Beate; Brysch, Wolfgang

Development of a Potent and Selective G2A (GPR132) Agonist.

开发一种高效选择性的G2A(GPR132)激动剂

Hernandez-Olmos Victor, Heering Jan, Marinescu Beatrice, Schermeng Tina, Ivanov Vladimir V, Moroz Yurii S, Nevermann Sheila, Mathes Marius, Ehrler Johanna H M, Alnouri Mohamad Wessam, Wolf Markus, Haydo Alicia S, Schmachtel Tessa, Zaliani Andrea, Höfner Georg, Kaiser Astrid, Schubert-Zsilavecz Manfred, Beck-Sickinger Annette G, Offermanns Stefan, Gribbon Philipp, Rieger Michael A, Merk Daniel, Sisignano Marco, Steinhilber Dieter, Proschak Ewgenij

Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation

靶向替代维生素E代谢物结合位点可实现非经典PPARγ调节

Arifi, Silvia; Marschner, Julian A; Pollinger, Julius; Isigkeit, Laura; Heitel, Pascal; Kaiser, Astrid; Obeser, Lennart; Höfner, Georg; Proschak, Ewgenij; Knapp, Stefan; Chaikuad, Apirat; Heering, Jan; Merk, Daniel