日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of an LSD1 PROTAC degrader.

发现一种LSD1 PROTAC降解酶

Hosseini Amir, Qiu Xing, Xiong Yan, Chiang Ki Him Nicholas, Catlett Jerrel, Kaltheuner Ines, Deng Zhijie, Ghosh Sudipta, Shi Yang, Jin Jian

Oncogenic CDK13 mutations impede nuclear RNA surveillance

致癌性 CDK13 突变会阻碍核 RNA 监视

Insco, Megan L; Abraham, Brian J; Dubbury, Sara J; Kaltheuner, Ines H; Dust, Sofia; Wu, Constance; Chen, Kevin Y; Liu, David; Bellaousov, Stanislav; Cox, Anna M; Martin, Benjamin J E; Zhang, Tongwu; Ludwig, Calvin G; Fabo, Tania; Modhurima, Rodsy; Esgdaille, Dakarai E; Henriques, Telmo; Brown, Kevin M; Chanock, Stephen J; Geyer, Matthias; Adelman, Karen; Sharp, Phillip A; Young, Richard A; Boutz, Paul L; Zon, Leonard I

Author Correction: LAMP-Seq enables sensitive, multiplexed COVID-19 diagnostics using molecular barcoding

作者更正:LAMP-Seq 利用分子条形码技术实现灵敏、多重 COVID-19 诊断。

Ludwig, Kerstin U; Schmithausen, Ricarda M; Li, David; Jacobs, Max L; Hollstein, Ronja; Blumenstock, Katja; Liebing, Jana; Słabicki, Mikołaj; Ben-Shmuel, Amir; Israeli, Ofir; Weiss, Shay; Ebert, Thomas S; Paran, Nir; Rüdiger, Wibke; Wilbring, Gero; Feldman, David; Lippke, Bärbel; Ishorst, Nina; Hochfeld, Lara M; Beins, Eva C; Kaltheuner, Ines H; Schmitz, Maximilian; Wöhler, Aliona; Döhla, Manuel; Sib, Esther; Jentzsch, Marius; Moench, Eva-Maria C; Borrajo, Jacob D; Strecker, Jonathan; Reinhardt, Julia; Cleary, Brian; Geyer, Matthias; Hölzel, Michael; Macrae, Rhiannon; Nöthen, Markus M; Hoffmann, Per; Exner, Martin; Regev, Aviv; Zhang, Feng; Schmid-Burgk, Jonathan L

Structure-activity relationship study of THZ531 derivatives enables the discovery of BSJ-01-175 as a dual CDK12/13 covalent inhibitor with efficacy in Ewing sarcoma

THZ531衍生物的构效关系研究发现了BSJ-01-175,它是一种对尤文氏肉瘤有效的双重CDK12/13共价抑制剂。

Jiang, Baishan; Jiang, Jie; Kaltheuner, Ines H; Iniguez, Amanda Balboni; Anand, Kanchan; Ferguson, Fleur M; Ficarro, Scott B; Seong, Bo Kyung Alex; Greifenberg, Ann Katrin; Dust, Sofia; Kwiatkowski, Nicholas P; Marto, Jarrod A; Stegmaier, Kimberly; Zhang, Tinghu; Geyer, Matthias; Gray, Nathanael S