Discovery of PXR Antagonist MI891 and PXR Degrader MI1013 and Their Roles in Hepatic Gene Regulation
PXR拮抗剂MI891和PXR降解剂MI1013的发现及其在肝脏基因调控中的作用
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c03134
Rajamanikkam Kamaraj ,Ivana Mejdrová ,Maria Krutakova ,Tomas Smutny ,Kryštof Škach ,Klara Dohnalova ,Lucie Smutna ,Dharani Sai Sreekanth Nellore ,Jan Dusek ,Karel Chalupsky ,Jana Hricová ,Thales Kronenberger ,Aaron Stahl ,Markus Templin ,Albert Braeuning ,Radim Nencka ,Petr Pavek