Discovery of Monovalent Direct Degraders of BRD4 that Act via the Recruitment of DCAF11
发现通过招募 DCAF11 发挥作用的 BRD4 单价直接降解剂
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-24-0219
Parker, Gregory S; Toth, Julia I; Fish, Sarah; Blanco, Gabrielle; Kampert, Taylor; Li, Xiaoming; Yang, Linette; Stumpf, Craig R; Steadman, Kenneth; Jamborcic, Aleksandar; Chien, Stephen; Daniele, Elizabeth; Dearie, Alejandro; Leriche, Geoffray; Bailey, Simon; Thompson, Peggy A