Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor
1-(5-氯-6-(三氟甲氧基)-1H-苯并咪唑-2-基)-1H-吡唑-4-羧酸(JNJ-42041935)的药理学表征,一种有效的选择性缺氧诱导因子脯氨酰羟化酶抑制剂
期刊:Molecular Pharmacology
影响因子:3.2
doi:10.1124/mol.110.070508
Terrance D Barrett, Heather L Palomino, Theresa I Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Peter V Haug, Wen Yan, Andrew Young, Hong Hua, Juliet C Hart, Da-Thao Tran, Hariharan Venkatesan, Mark D Rosen, Hillary M Peltier, Kia Sepassi, Michele C Rizzolio, Scott D Bembenek, Tara Mirzadegan, Micha