日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Time-resolved spectroscopy of a photoactive dinuclear W/Ru complex: spectroscopic evidence for a metastable intermediate with side-on coordinated carbonyl ligand

光活性双核W/Ru配合物的时间分辨光谱:具有侧向配位羰基配体的亚稳态中间体的光谱证据

Borter, Jan-Hendrik; Kangsa Banik, Sayan; Kunze, Kristian; Kupfer, Stephan; Schwarzer, Dirk; Seidel, Wolfram W

Discovery of Fragment-Based Inhibitors of SARS-CoV-2 PL(Pro)

SARS-CoV-2 PL(Pro)片段抑制剂的发现

Wei, Qiangqiang; Taylor, Ashley J; Barmade, Mahesh Angadrao; Teuscher, Kevin B; Chowdhury, Somanath; Apakama, Chideraa; Anderson-Daniels, Jordan; Yongqing, Zhu; Schultz, David C; Rietz, Tyson A; South, Taylor M; Crow, Mackenzie M; Zhao, Bin; Amporndanai, Kangsa; Sensintaffar, John L; Phan, Jason; Cherry, Sara; Denison, Mark; Lee, Taekyu; Fesik, Stephen W

Discovery of Spiro[chromane-2,4'-piperidine] Derivatives as Irreversible Inhibitors of SARS-CoV-2 Papain-like Protease

发现螺[色满-2,4'-哌啶]衍生物作为SARS-CoV-2木瓜蛋白酶样蛋白酶的不可逆抑制剂

Wei, Qiangqiang; Taylor, Ashley J; Miriyala, Nagaraju; Barmade, Mahesh A; Gentry, Zachary O; Anderson-Daniels, Jordan; Teuscher, Kevin B; Crow, Mackenzie M; Apakama, Chideraa; South, Taylor M; Rietz, Tyson A; Amporndanai, Kangsa; Phan, Jason; Sensintaffar, John L; Denison, Mark; Lee, Taekyu; Fesik, Stephen W

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

Cooperativity of Electron Transfer Coupled Spin Transitions in a Tetranuclear Fe/Co Prussian Blue Analogue Revealed by Ultrafast Spectroscopy

超快光谱揭示四核铁/钴普鲁士蓝类似物中电子转移耦合自旋转变的协同性

Borter, Jan-Hendrik; Kar, Simindokht Gol; Kangsa Banik, Sayan; Demeshko, Serhiy; Oswald, Rainer; Gimferrer, Martí; Mata, Ricardo A; Schwarzer, Dirk; Meyer, Franc

Nuclear Magnetic Resonance-based fragment screen of the E3 ligase Fem-1 homolog B

基于核磁共振的E3连接酶Fem-1同源物B片段筛选

Katinas, Jade M; Amporndanai, Kangsa; Taylor, Ashley J; Rose, Kristie L; Gareiss, Peter C; Crespo, Roberto A; Phan, Jason; Waterson, Alex G; Fesik, Stephen W

NMR-Based Fragment Screen of the von Hippel-Lindau Elongin C&B Complex

基于核磁共振的von Hippel-Lindau Elongin C&B复合物片段筛选

Amporndanai, Kangsa; Katinas, Jade M; Chopra, Ashima; Kayode, Olumide; Vadukoot, Anish K; Waterson, Alex G; Fesik, Stephen W

Fragment-Based Screen of SARS-CoV-2 Papain-like Protease (PL(pro))

基于片段的SARS-CoV-2木瓜蛋白酶样蛋白酶(PL(pro))筛选

Taylor, Ashley J; Amporndanai, Kangsa; Rietz, Tyson A; Zhao, Bin; Thiruvaipati, Anusha; Wei, Qiangqiang; South, Taylor M; Crow, Mackenzie M; Apakama, Chideraa; Sensintaffar, John L; Phan, Jason; Lee, Taekyu; Fesik, Stephen W

Ebselen analogues delay disease onset and its course in fALS by on-target SOD-1 engagement

依布硒啉类似物通过靶向SOD-1受体,延缓fALS的发病和病程。

Seiji Watanabe # ,Kangsa Amporndanai # ,Raheela Awais # ,Caroline Latham ,Muhammad Awais ,Paul M O'Neill ,Koji Yamanaka ,S Samar Hasnain

Targeting the Ubiquinol-Reduction (Q(i)) Site of the Mitochondrial Cytochrome bc(1) Complex for the Development of Next Generation Quinolone Antimalarials

靶向线粒体细胞色素bc(1)复合物的泛醌还原(Q(i))位点以开发下一代喹诺酮类抗疟药

Amporndanai, Kangsa; Pinthong, Nattapon; O'Neill, Paul M; Hong, W David; Amewu, Richard K; Pidathala, Chandrakala; Berry, Neil G; Leung, Suet C; Ward, Stephen A; Biagini, Giancarlo A; Hasnain, S Samar; Antonyuk, Svetlana V