日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

发现一种可调节小鼠情绪行为的 NAPE-PLD 抑制剂

Elliot D Mock, Mohammed Mustafa, Ozge Gunduz-Cinar, Resat Cinar, Gavin N Petrie, Vasudev Kantae, Xinyu Di, Daisuke Ogasawara, Zoltan V Varga, Janos Paloczi, Cristina Miliano, Giulia Donvito, Annelot C M van Esbroeck, Anouk M F van der Gracht, Ioli Kotsogianni, Joshua K Park, Andrea Martella, Tom van

Structure-Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family

α-酮酰胺作为磷脂酶 A 和酰基转移酶家族抑制剂的构效关系研究

Juan Zhou, Elliot D Mock, Karol Al Ayed, Xinyu Di, Vasudev Kantae, Lindsey Burggraaff, Anna F Stevens, Andrea Martella, Florian Mohr, Ming Jiang, Tom van der Wel, Tiemen J Wendel, Tim P Ofman, Yvonne Tran, Nicky de Koster, Gerard J P van Westen, Thomas Hankemeier, Mario van der Stelt

Impact of post-hatching maturation on the pharmacokinetics of paracetamol in zebrafish larvae

孵化后成熟对斑马鱼幼体中对乙酰氨基酚药代动力学的影响

van Wijk, Rob C; Krekels, Elke H J; Kantae, Vasudev; Harms, Amy C; Hankemeier, Thomas; van der Graaf, Piet H; Spaink, Herman P

Activity-Based Protein Profiling Identifies α-Ketoamides as Inhibitors for Phospholipase A2 Group XVI

基于活性的蛋白质谱分析鉴定出α-酮酰胺是磷脂酶A2第十六组的抑制剂

Zhou, Juan; Mock, Elliot D; Martella, Andrea; Kantae, Vasudev; Di, Xinyu; Burggraaff, Lindsey; Baggelaar, Marc P; Al-Ayed, Karol; Bakker, Alexander; Florea, Bogdan I; Grimm, Sebastian H; den Dulk, Hans; Li, Chun T; Mulder, Laura; Overkleeft, Herman S; Hankemeier, Thomas; van Westen, Gerard J P; van der Stelt, Mario

Identification of α,β-Hydrolase Domain Containing Protein 6 as a Diacylglycerol Lipase in Neuro-2a Cells

鉴定含 α,β-水解酶结构域的蛋白 6 为 Neuro-2a 细胞中的二酰甘油脂肪酶

Annelot C M van Esbroeck, Vasudev Kantae, Xinyu Di, Tom van der Wel, Hans den Dulk, Anna F Stevens, Simar Singh, Alexander T Bakker, Bogdan I Florea, Nephi Stella, Herman S Overkleeft, Thomas Hankemeier, Mario van der Stelt

Caloric restriction lowers endocannabinoid tonus and improves cardiac function in type 2 diabetes

热量限制可降低内源性大麻素张力并改善2型糖尿病患者的心脏功能

van Eyk, Huub J; van Schinkel, Linda D; Kantae, Vasudev; Dronkers, Charlotte E A; Westenberg, Jos J M; de Roos, Albert; Lamb, Hildo J; Jukema, J Wouter; Harms, Amy C; Hankemeier, Thomas; van der Stelt, Mario; Jazet, Ingrid M; Rensen, Patrick C N; Smit, Johannes W A

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474

基于活性的蛋白质谱分析揭示了FAAH抑制剂BIA 10-2474的脱靶蛋白

van Esbroeck, Annelot C M; Janssen, Antonius P A; Cognetta, Armand B 3rd; Ogasawara, Daisuke; Shpak, Guy; van der Kroeg, Mark; Kantae, Vasudev; Baggelaar, Marc P; de Vrij, Femke M S; Deng, Hui; Allarà, Marco; Fezza, Filomena; Lin, Zhanmin; van der Wel, Tom; Soethoudt, Marjolein; Mock, Elliot D; den Dulk, Hans; Baak, Ilse L; Florea, Bogdan I; Hendriks, Giel; De Petrocellis, Luciano; Overkleeft, Herman S; Hankemeier, Thomas; De Zeeuw, Chris I; Di Marzo, Vincenzo; Maccarrone, Mauro; Cravatt, Benjamin F; Kushner, Steven A; van der Stelt, Mario

Quantitative profiling of endocannabinoids and related N-acylethanolamines in human CSF using nano LC-MS/MS

使用纳米 LC-MS/MS 对人类脑脊液中的内源性大麻素和相关 N-酰基乙醇胺进行定量分析

Vasudev Kantae, Shinji Ogino, Marek Noga, Amy C Harms, Robin M van Dongen, Gerrit L J Onderwater, Arn M J M van den Maagdenberg, Gisela M Terwindt, Mario van der Stelt, Michel D Ferrari, Thomas Hankemeier

Endocannabinoid tone is higher in healthy lean South Asian than white Caucasian men

健康瘦弱的南亚男性的内源性大麻素水平高于白种人男性

Vasudev Kantae, Kimberly J Nahon, Maaike E Straat, Leontine E H Bakker, Amy C Harms, Mario van der Stelt, Thomas Hankemeier, Ingrid M Jazet, Mariëtte R Boon, Patrick C N Rensen

Integration of pharmacometabolomics with pharmacokinetics and pharmacodynamics: towards personalized drug therapy

将药物代谢组学与药代动力学和药效学相结合:迈向个体化药物治疗

Kantae, Vasudev; Krekels, Elke H J; Esdonk, Michiel J Van; Lindenburg, Peter; Harms, Amy C; Knibbe, Catherijne A J; Van der Graaf, Piet H; Hankemeier, Thomas