日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Microbial Cross-Talk: Unlocking the Cytochalasin Diversity from a Termite-Associated Xylaria

微生物间的相互作用:揭示白蚁相关木霉属真菌细胞松弛素的多样性

Dayras, Marie; Liu, Yaming; Kochems, Rebecca; de Kruijff, Martinus; Balluff, Sven; Rasheed, Sari; Kany, Andreas M; Herrmann, Jennifer; Götze, Sebastian; Morgenstern, Bernd; Koné, N'Golo A; Poulsen, Michael; Müller, Rolf; Beemelmanns, Christine

Multiparameter Optimization of Pseudomonas aeruginosa Elastase Inhibitors for Systemic Administration

铜绿假单胞菌弹性蛋白酶抑制剂全身给药的多参数优化

Abdelsamie, Ahmed S; Konstantinović, Jelena; Kany, Andreas M; Schütz, Christian; Kolling, Dominik; Speicher, Samira; Klein, Andreas; Shafiei, Roya; Bouté, Mélodie; Mundry, Katharina; Park, Yu Mi; Loretz, Brigitta; Müller, Rolf; Sallenave, Jean-Michel; Lehr, Claus-Michael; Koehnke, Jesko; Rox, Katharina; Haupenthal, Jörg; Hirsch, Anna K H

Structure Elucidation, Biosynthesis and Biological Evaluation of Neosorangicin A, a Member of the Sorangicin Family

新索兰吉辛A(索兰吉辛家族成员)的结构解析、生物合成及生物学评价

Fries, Franziska; Walesch, Sebastian; Jansen, Rolf; von Peinen, Kristin; Mehr, Luisa; Pätzold, Linda; Karwehl, Sabrina; Kany, Andreas M; Garcia, Ronald; Reinecke, Silke; Haupenthal, Jörg; Stradal, Theresia E B; Bischoff, Markus; Stadler, Marc; Müller, Rolf; Herrmann, Jennifer

Dipeptidic Phosphonates: Potent Inhibitors of Pseudomonas aeruginosa Elastase B Showing Efficacy in a Murine Keratitis Model

二肽膦酸酯:铜绿假单胞菌弹性蛋白酶B的强效抑制剂,在小鼠角膜炎模型中显示出疗效

Kiefer, Alexander F; Schütz, Christian; Englisch, Colya N; Kolling, Dominik; Speicher, Samira; Kany, Andreas M; Shafiei, Roya; Wadood, Noran A; Aljohmani, Ahmad; Wirschem, Niklas; Jumde, Ravindra P; Klein, Andreas; Sikandar, Asfandyar; Park, Yu-Mi; Krasteva-Christ, Gabriela; Yildiz, Daniela; Abdelsamie, Ahmed S; Rox, Katharina; Köhnke, Jesko; Müller, Rolf; Bischoff, Markus; Haupenthal, Jörg; Hirsch, Anna K H

Engineering an Artificial Myxopyronin Derivative with Enhanced Metabolic Stability via Mutasynthesis

通过突变合成工程构建具有增强代谢稳定性的人工粘液吡喃酮衍生物

Kiefer, Alexander F; Voltz, Alexander; Scherzer, Domen; Reberšek, Roman; Kany, Andreas M; Prosser, Gareth; Neuber, Markus; Reiling, Norbert; Hirsch, Anna K H; Müller, Rolf

Tailored phenyl ureas eradicate drug-resistant Mycobacterium tuberculosis by targeting mycolic acid cell wall assembly

定制的苯脲类化合物通过靶向分枝菌酸细胞壁组装来根除耐药结核分枝杆菌。

Mostert, Dietrich; Braun, Josef; Zimmerman, Matthew D; Engelhart, Curtis A; Berndl, Sara; Quoika, Patrick K; Kany, Andreas M; Proietto, Julianna; Penalva-Lopez, Suyapa; Wallach, Joshua B; Hirsch, Anna K H; Zacharias, Martin; Schnappinger, Dirk; Dartois, Véronique; Sieber, Stephan A

Design, Synthesis, and Biological Evaluation of Mono- and Diamino-Substituted Squaramide Derivatives as Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthase

单氨基和二氨基取代的方酰胺衍生物作为结核分枝杆菌腺苷三磷酸(ATP)合成酶的强效抑制剂的设计、合成和生物学评价

Palme, Paul R; Grover, Shipra; Abdelaziz, Rana; Mann, Lea; Kany, Andreas M; Ouologuem, Lina; Bartel, Karin; Sonnenkalb, Lindsay; Reiling, Norbert; Hirsch, Anna K H; Schnappinger, Dirk; Rubinstein, John L; Imming, Peter; Richter, Adrian

Structure Revision of Halisphingosine A via Total Synthesis and Bioactivity Studies

通过全合成和生物活性研究对哈利鞘氨醇A的结构进行修正

Sauer, Maria; Kany, Andreas M; Götze, Sebastian; Müller, Rolf; Beemelmanns, Christine

Isocyanides inhibit bacterial pathogens by covalent targeting of essential metabolic enzymes

异氰化物通过共价靶向必需代谢酶来抑制细菌病原体。

Geißler, Alexandra; Junca, Howard; Kany, Andreas M; Daumann, Lena J; Hirsch, Anna K H; Pieper, Dietmar H; Sieber, Stephan A

Thermo-amplifier circuit in probiotic E. coli for stringently temperature-controlled release of a novel antibiotic.

利用益生菌大肠杆菌中的热放大器电路,严格控制温度释放新型抗生素

Dey Sourik, Seyfert Carsten E, Fink-Straube Claudia, Kany Andreas M, Müller Rolf, Sankaran Shrikrishnan