日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

LYMTACs:chimeric small molecules repurpose lysosomal membrane proteins for target protein relocalization and degradation.

LYMTACs:嵌合小分子可重新利用溶酶体膜蛋白,实现靶蛋白的重新定位和降解

Nalawansha Dhanusha A, Mazis Georgios, Husemoen Gitte, Ashton Kate S, Deng Weixian, Wurz Ryan P, Tran Anh T, Lanman Brian A, Xie Jiansong, Guenette Robert G, Li Shiqian, Smith Christopher E, Archunan Suresh, Agnihotram Manoj K, Sadhukhan Arghya, Kapoor Rajiv, Wilde Chris, Koirala Sajjan, De Sousa E Melo Felipe, Potts Patrick Ryan

From DNA-Encoded Library Screening to AM-9747: An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo Efficacy.

从 DNA 编码文库筛选到 AM-9747:一种具有强效口服体内疗效的 MTA 协同 PRMT5 抑制剂

Sarvary Ian, Vestergaard Mikkel, Moretti Loris, Andersson Jan, Peiró Cadahía Jorge, Cowland Sanne, Flagstad Thomas, Franch Thomas, Gouliaev Alex, Husemoen Gitte, Jacso Tomas, Kronborg Titi, Kuropatnicka Aleksandra, Nadali Anna, Madsen Mads, Nielsen So Ren, Pii David, Ryborg So Ren, Soede Camillia, Allen Jennifer R, Bourbeau Matthew, Li Kexue, Liu Qingyian, Lo Mei-Chu, Madoux Franck, Mardirossian Narbe, Moriguchi Jodi, Ngo Rachel, Peng Chi-Chi, Pettus Liping, Tamayo Nuria, Wang Paul, Kapoor Rajiv, Belmontes Brian, Caenepeel Sean, Hughes Paul, Liu Siyuan, Slemmons Katherine K, Yang Yajing, Xie Fang, Ghimire-Rijal Sudipa, Mukund Susmith, Glad Sanne

MRI-Derived Fat Fraction Is Superior to Ultrasonography in Predicting Subclinical Atherosclerosis in Metabolically Healthy Non-alcoholic Fatty Liver Disease

磁共振成像衍生的脂肪分数在预测代谢健康非酒精性脂肪肝患者的亚临床动脉粥样硬化方面优于超声检查

Bhawariya, Sunil; Bhardwaj, Arshia; Singh, Arshdeep; Sharma, Riya; Kapoor, Rajiv; Bawa, Ashutosh; Joshi, Liza; Bhardwaj, Gopal