日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CDK/mTOR-dependent phosphorylation of UBE2H restrains its charging with ubiquitin and regulates CTLH-dependent degradation

UBE2H的CDK/mTOR依赖性磷酸化抑制其泛素化,并调节CTLH依赖性降解。

Chen, Yingqian; Rossio, Valentina; Paulo, Joao A; Karki, Menuka; Manohar, Sandhya; Ozimek, Noelle; Frizzi, Laura; Gygi, Steven P; King, Randall W

Lysine Demethylase 4A (KDM4A) Maintains Basal Body Architecture and Protects Against Ciliary Destabilization

赖氨酸去甲基酶4A (KDM4A) 维持基体结构并防止纤毛不稳定

Motrapu, Manga; Hudson, Lindsey; Chowdhury, Pratim; Wang, Xiaoli; Nakatani, Yuya; Vargas-Hernandez, Sofia; Jung, Sung Y; Karki, Menuka; Walker, Cheryl; Gustavsson, Anna-Karin; Dere, Ruhee

Sitravatinib in combination with nivolumab plus ipilimumab in patients with advanced clear cell renal cell carcinoma: a phase 1 trial

西曲替尼联合纳武利尤单抗和伊匹木单抗治疗晚期透明细胞肾细胞癌患者:一项 I 期试验

Msaouel, Pavlos; Yu, Kai; Yuan, Ying; Chen, Jianfeng; Yan, Xinmiao; Karki, Menuka; Duan, Fei; Sheth, Rahul A; Rao, Priya; Sircar, Kanishka; Shah, Amishi Y; Zurita, Amado J; Genovese, Giannicola; Li, Min; Yeh, Chih-Chen; Dang, Minghao; Han, Guangchun; Chu, Yanshuo; Hallin, Max; Olson, Peter; Yang, Rui; Slavin, Daniela; Der-Torossian, Hirak; Chin, Curtis D; Tannir, Nizar M; Wang, Linghua; Gao, Jianjun

Nivolumab plus ipilimumab induce hyper-progression in renal medullary carcinoma: results of a phase II trial and preclinical evidence.

纳武利尤单抗联合伊匹木单抗可诱导肾髓质癌超进展:II期试验结果和临床前证据。

Soeung Melinda, Yan Xinmiao, Zanca Ciro, Qian Jing, Karki Menuka, Duan Fei, Khan Hania, Zhang Li, Peng David H, Williams Mariah, He Rong, Chen Ziheng, Perelli Luigi, Chen Jianfeng, Tidwell Rebecca S, Chauhan Pankaj K, Le Courtney N, Lam Truong N A, Bhattacharya Nirjar, Shah Rutvi, Ho I-Lin, Gay Jason P, Carrillo Caroline C, Feng Ningping, Le Kang, Gao Guang, Perry Teresa L, Mseeh Faika, Jiang Yongying, Xu Quanyun A, Zacharias Niki Marie, Sheth Rahul A, Bathala Tharakeswara K, Rao Priya, Daw Najat C, Tripathi Durga N, Walker Cheryl L, Mohammad Mohammad M, Zhang Jianhua, Han Guangchun, Chu Yanshuo, Wang Ruiping, Dang Minghao, Dai Enyu, Peng Fuduan, Liu Yunhe, Jadhav Akshaya, Lang Wenhua, Arrechedera Claudio A, Clemente Leticia Campos, Parra Edwin R, Lu Hsinyi, Haymaker Cara L, Wistuba Ignacio I, Futreal Andrew, Viale Andrea, Soth Michael J, Jones Philip, Marszalek Joseph R, Heffernan Timothy, Draetta Giulio F, Tannir Nizar M, Gao Jianjun, Wang Linghua, Genovese Giannicola, Msaouel Pavlos

Identification of therapeutic targets for renal medullary carcinoma via integrated genomic and transcriptomic profiling.

通过整合基因组和转录组分析鉴定肾髓质癌的治疗靶点。

Msaouel Pavlos, Tannir Nizar M, Meric-Bernstam Funda, King Jennifer M, Voss Martin H, Cheng Jessica P, Thomas Susan S, Lim Zita D, Karki Menuka, He Rong, Genovese Giannicola, Sheth Rahul A, Ingram Davis R, Shamsutdinova Diana, Wani Khalida M, Wang Wei-Lien, Lazar Alexander J, Knipper-Davis Dominique, Berlinski Amber, Soares Tayla, Stupichev Danil, Kryukov Kirill, Davitavyan Suren, Novokreshchenova Anna, Lebedev Dmitry, Kurpe Stanislav, Kravets Andrey, Belousov Dmitrii, Hensley Michael, Bagaev Alexander, Paradiso Francesca, Kushnarev Vladimir

CA-125 as a Biomarker in Renal Medullary Carcinoma: Integrated Molecular Profiling, Functional Characterization, and Prospective Clinical Validation.

CA-125 作为肾髓质癌的生物标志物:整合分子谱分析、功能表征和前瞻性临床验证

Grimm Sandra L, Karki Menuka, Blum Kyle A, Bertocchio Jean-Philippe, He Rong, Tripathi Durga N, Zacharias Niki M, Lebenthal Justin M, Sheth Rahul A, Rao Priya, Genovese Giannicola, Lu Zhen, Bast Robert C, Ingram Davis R, Lazcano Rossana, Wani Khalida M, Wang Wei-Lien, Lazar Alexander J, Tannir Nizar M, Walker Cheryl L, Coarfa Cristian, Msaouel Pavlos

Differential Efficacy of Bevacizumab and Erlotinib in Preclinical Models of Renal Medullary Carcinoma and Fumarate Hydratase-Deficient Renal Cell Carcinoma.

贝伐珠单抗和厄洛替尼在肾髓质癌和富马酸水合酶缺乏型肾细胞癌临床前模型中的差异疗效

Zacharias Niki M, Ozambela Manuel, Karki Menuka, He Rong, Chauhan Pankaj K, Pesquera Pedro I, Hernandez Gonzalez Andres E, Ochoa Oscar, Pieretti Alberto, Chen Huiqin, De La Cerda Carolyn, Yu Zhiyuan, Grover Abha, Hicks-Peña Samantha, Fowlkes Natalie W, Wang Lei, Maity Tapati, Rao Priya, Genovese Giannicola, Tannir Nizar M, Karam Jose A, Msaouel Pavlos

Neuronal SETD2 activity links microtubule methylation to an anxiety-like phenotype in mice

神经元SETD2活性将微管甲基化与小鼠的焦虑样表型联系起来

Koenning, Matthias; Wang, Xianlong; Karki, Menuka; Jangid, Rahul Kumar; Kearns, Sarah; Tripathi, Durga Nand; Cianfrocco, Michael; Verhey, Kristen J; Jung, Sung Yun; Coarfa, Cristian; Ward, Christopher Scott; Kalish, Brian Thomas; Grimm, Sandra L; Rathmell, W Kimryn; Mostany, Ricardo; Dere, Ruhee; Rasband, Matthew Neil; Walker, Cheryl Lyn; Park, In Young

Synthetic and biological studies of tubulin targeting c2-substituted 7-deazahypoxanthines derived from marine alkaloid rigidins

对源自海洋生物碱刚毛素的 C2 位取代的 7-脱氮次黄嘌呤类化合物进行合成和生物学研究,这些化合物靶向微管蛋白。

Scott, Robert; Karki, Menuka; Reisenauer, Mary R; Rodrigues, Roberta; Dasari, Ramesh; Smith, W Ross; Pelly, Stephen C; van Otterlo, Willem A L; Shuster, Charles B; Rogelj, Snezna; Magedov, Igor V; Frolova, Liliya V; Kornienko, Alexander

Exploring natural product chemistry and biology with multicomponent reactions. 5. Discovery of a novel tubulin-targeting scaffold derived from the rigidin family of marine alkaloids

利用多组分反应探索天然产物化学和生物学。5. 发现一种源自海洋生物碱刚毛素家族的新型微管蛋白靶向支架。

Frolova, Liliya V; Magedov, Igor V; Romero, Anntherese E; Karki, Menuka; Otero, Isaiah; Hayden, Kathryn; Evdokimov, Nikolai M; Banuls, Laetitia Moreno Y; Rastogi, Shiva K; Smith, W Ross; Lu, Shi-Long; Kiss, Robert; Shuster, Charles B; Hamel, Ernest; Betancourt, Tania; Rogelj, Snezna; Kornienko, Alexander