日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Novel JAK2 Inhibitors from Amino Derivatives of Epoxyalantolactone: In Silico and In Vitro Studies

从环氧阿兰内酯氨基衍生物中鉴定新型JAK2抑制剂:计算机模拟和体外研究

Todsaporn, Duangjai; Sanachai, Kamonpan; Aonbangkhen, Chanat; Poo-Arporn, Rungtiva P; Kartsev, Victor; Pukhov, Sergey; Afanasyeva, Svetlana; Geronikaki, Athina; Rungrotmongkol, Thanyada

Investigating Amphoteric 3,4'-Biscoumarin-Based ortho-[(Dialkylamino)methyl]phenols as Dual MAO and ChE Inhibitors

研究两性3,4'-双香豆素基邻-[(二烷基氨基)甲基]苯酚作为MAO和ChE双重抑制剂

Petrou, Anthi; Deruvo, Caterina; Purgatorio, Rosa; Lichitsky, Boris; Komogortsev, Andrey N; Kartsev, Victor G; de Candia, Modesto; Catto, Marco; Altomare, Cosimo D; Geronikaki, Athina

Exploring novel furochochicine derivatives as promising JAK2 inhibitors in HeLa cells: Integrating docking, QSAR-ML, MD simulations, and experiments.

探索新型呋喃妥因衍生物作为 HeLa 细胞中 JAK2 抑制剂的潜力:整合对接、QSAR-ML、MD 模拟和实验

Todsaporn Duangjai, Sanachai Kamonpan, Aonbangkhen Chanat, Geronikaki Athina, Kartsev Victor, Lichitsky Boris, Komogortsev Andrey, Maitarad Phornphimon, Rungrotmongkol Thanyada

A Universal Method for the Synthesis of new Heterocyclic Systems: Pyrimido[2,1-f][1,2,4]triazines

一种合成新型杂环体系的通用方法:嘧啶并[2,1-f][1,2,4]三嗪

Sirakanyan, Samvel N; Spinelli, Domenico; Geronikaki, Athina; Kartsev, Victor G; Hakobyan, Elmira K; Jughetsyan, Hasmik V; Yegoryan, Hasmik A; Hovakimyan, Anush A

Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors

灰黄霉素和地衣酸磺酰胺衍生物作为真菌、细菌和人类碳酸酐酶抑制剂的合成、生物学和计算机模拟研究

Angeli, Andrea; Petrou, Anthi; Kartsev, Victor; Lichitsky, Boris; Komogortsev, Andrey; Capasso, Clemente; Geronikaki, Athina; Supuran, Claudiu T

Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives

5-吲哚基亚甲基-4-氧代-2-硫代噻唑烷衍生物的合成、生物学评价和分子对接研究

Horishny, Volodymyr; Geronikaki, Athina; Kartsev, Victor; Matiychuk, Vasyl; Petrou, Anthi; Pogodin, Pavel; Poroikov, Vladimir; Papadopoulou, Theodora A; Vizirianakis, Ioannis S; Kostic, Marina; Ivanov, Marija; Sokovic, Marina

Synthesis and Antimicrobial Activity of New Heteroaryl(aryl) Thiazole Derivatives Molecular Docking Studies

新型杂芳基(芳基)噻唑衍生物的合成及其抗菌活性分子对接研究

Kartsev, Victor; Geronikaki, Athina; Zubenko, Alexander; Petrou, Anthi; Ivanov, Marija; Glamočlija, Jasmina; Sokovic, Marina; Divaeva, Lyudmila; Morkovnik, Anatolii; Klimenko, Alexander

Experimental and In Silico Evaluation of New Heteroaryl Benzothiazole Derivatives as Antimicrobial Agents

新型杂芳基苯并噻唑衍生物作为抗菌剂的实验和计算机模拟评价

Zubenko, Alexander; Kartsev, Victor; Petrou, Anthi; Geronikaki, Athina; Ivanov, Marija; Glamočlija, Jasmina; Soković, Marina; Divaeva, Lyudmila; Morkovnik, Anatolii; Klimenko, Alexander

Disruption of the Complex between GAPDH and Hsp70 Sensitizes C6 Glioblastoma Cells to Hypoxic Stress

GAPDH与Hsp70复合物的破坏使C6胶质母细胞瘤细胞对缺氧应激更加敏感

Mikeladze, Marina A; Dutysheva, Elizaveta A; Kartsev, Victor G; Margulis, Boris A; Guzhova, Irina V; Lazarev, Vladimir F

Synthesis and Neurotropic Activity of New Heterocyclic Systems: Pyridofuro[3,2-d]pyrrolo[1,2-a]pyrimidines, Pyridofuro[3,2-d]pyrido[1,2-a]pyrimidines and Pyridofuro[3',2':4,5]pyrimido[1,2-a]azepines

新型杂环体系的合成及神经活性:吡啶呋喃并[3,2-d]吡咯并[1,2-a]嘧啶、吡啶呋喃并[3,2-d]吡啶并[1,2-a]嘧啶和吡啶呋喃并[3',2':4,5]嘧啶并[1,2-a]氮杂环庚烷

Sirakanyan, Samvel N; Spinelli, Domenico; Geronikaki, Athina; Kartsev, Victor; Hakobyan, Elmira K; Petrou, Anthi; Paronikyan, Ruzanna G; Nazaryan, Ivetta M; Akopyan, Hasmik H; Hovakimyan, Anush A